SCHEMBL8587367

SCHEMBL8587367

COc1nc(N)nc2c1ncn2[C@@H]1O[C@H](CO)[C@](O)(C(C)=O)[C@@]1(O)C(C)=O

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.41
CYP2C19 P33261 1/20 0.38
ADORA3 P0DMS8 2/20 0.37
ADORA1 P30542 2/20 0.37
ADORA2B P29275 2/20 0.37
ADA P00813 1/20 0.36
HSP90B1 P14625 1/20 0.36
SLC29A1 Q99808 4/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
HINT1 P49773 1/20 0.35
PGK1 P00558 1/20 0.34
PGK2 P07205 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16125688 0.83 ADORA2A (0.45) ADORA2ACYP2C19ADORA3ADORA1ADORA2B
SCHEMBL8587151 0.83 ADORA3 (0.35) ADORA2AADORA3ADORA1ADORA2BHSP90B1
SCHEMBL31293603 0.79 ADORA3 (0.47) ADORA3HINT1
SCHEMBL3622556 0.79 ADORA2A (0.59) ADORA2AADORA3ADORA1ADORA2BADA
Beta-2'-C-Methyl-6-O-Methyl Guanosine SCHEMBL12939406 0.78 ADORA2A (0.66) ADORA2ACYP2C19ADORA3ADORA1ADORA2B
Beta-2'-C-Methyl-6-O-Methyl Guanosine SCHEMBL15628197 0.78 ADORA2A (0.66) ADORA2ACYP2C19ADORA3ADORA1ADORA2B
Beta-2'-C-Methyl-6-O-Methyl Guanosine SCHEMBL14762374 0.78 ADORA2A (0.66) ADORA2ACYP2C19ADORA3ADORA1ADORA2B
Beta-2'-C-Methyl-6-O-Methyl Guanosine SCHEMBL14816756 0.78 ADORA2A (0.66) ADORA2ACYP2C19ADORA3ADORA1ADORA2B
Beta-2'-C-Methyl-6-O-Methyl Guanosine SCHEMBL19493379 0.78 ADORA2A (0.66) ADORA2ACYP2C19ADORA3ADORA1ADORA2B
Beta-2'-C-Methyl-6-O-Methyl Guanosine SCHEMBL12219172 0.78 ADORA2A (0.66) ADORA2ACYP2C19ADORA3ADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992001456-A1 HETEROCYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1992-02-06 WO claimed
WO-1998042352-A1 METHOD FOR TREATING B-CELL TUMORS WITH ARA-G NUCLEOSIDE DERIVATIVES GLAXO GROUP LTD. (GB) 1998-10-01 WO disclosed
WO-1992001456-A1 HETEROCYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1992-02-06 WO disclosed