SCHEMBL8587151

SCHEMBL8587151

COc1nc(N)nc2c1ncn2[C@@H]1O[C@H](C(O)C(C)=O)[C@](O)(C(C)=O)[C@@]1(O)C(C)=O

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 8/20 0.35
ADORA2B P29275 8/20 0.35
ADORA1 P30542 8/20 0.35
ADORA2A P29274 6/20 0.34
HSP90B1 P14625 1/20 0.33
HINT1 P49773 1/20 0.33
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
NT5E P21589 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5492971 0.87 NT5E (0.38) ADORA3ADORA2BADORA1ADORA2AHSP90B1
SCHEMBL9791026 0.85 ADORA3 (0.35) ADORA3ADORA2BADORA1ADORA2AHSP90B1
SCHEMBL8587367 0.83 ADORA2A (0.41) ADORA3ADORA2BADORA1ADORA2AHSP90B1
SCHEMBL8588710 0.82 ADORA3 (0.38) ADORA3ADORA2BADORA1ADORA2AHSP90B1
SCHEMBL8588424 0.82 ADORA3 (0.42) ADORA3ADORA2BADORA1ADORA2AHSP90B1
SCHEMBL1120685 0.80 HINT1 (0.43) ADORA3HINT1
SCHEMBL30544925 0.79 ADORA2A (0.49) ADORA3ADORA2BADORA1ADORA2AHSP90B1
SCHEMBL4948918 0.79 LMNA (0.43) ADORA3ADORA2BADORA1ADORA2ANT5E
SCHEMBL1433825 0.78 DNMT1 (0.39)
SCHEMBL5498228 0.78 LMNA (0.37) ADORA3ADORA2BADORA1ADORA2ANT5E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992001456-A1 HETEROCYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1992-02-06 WO claimed
WO-1998042352-A1 METHOD FOR TREATING B-CELL TUMORS WITH ARA-G NUCLEOSIDE DERIVATIVES GLAXO GROUP LTD. (GB) 1998-10-01 WO disclosed
WO-1992001456-A1 HETEROCYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1992-02-06 WO disclosed