SCHEMBL8588798

SCHEMBL8588798

Nn1c[c]c2ccccc21

nearest known ligand 0.31

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
THPO P40225 1/20 0.31
CYP4Z1 Q86W10 1/20 0.31
NOS2 P35228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL193935 0.71 GPR3 (0.37) ALDH1A1MAPT
SCHEMBL5373174 0.71 KDM4E (0.34)
SCHEMBL7288679 0.71
SCHEMBL9581901 0.69 BCHE (0.35) CYP3A4MAPT
SCHEMBL4014977 0.67 L3MBTL1 (0.38) ALDH1A1CYP1A2MAPT
SCHEMBL9581979 0.67
SCHEMBL10813815 0.67
SCHEMBL3054238 0.67 EGFR (0.30)
SCHEMBL2268788 0.67 SMN1; SMN2 (0.38) ALDH1A1
SCHEMBL405536 0.67 TSHR (0.33) ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483881-B1 3-Amidoindolyl derivatives MERRELL PHARMA INC (US) 1998-01-21 EP disclosed
EP-0483881-A1 3-Amidoindolyl derivatives MERRELL PHARMACEUTICALS INC. (US) 1992-05-06 EP disclosed