SCHEMBL8589503

SCHEMBL8589503

O=c1[nH]c2cc(C(F)(F)F)c([N+](=O)[O-])cc2n(Nc2ccccc2)c1=O

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.47
CA9 Q16790 1/20 0.47
PARP1 P09874 1/20 0.46
GRIK1 P39086 6/20 0.45
GRIA1 P42261 6/20 0.45
GRIA2 P42262 6/20 0.45
GRIA3 P42263 6/20 0.45
GRIA4 P48058 6/20 0.45
GRIK2 Q13002 6/20 0.45
GRIK3 Q13003 6/20 0.45
GRIK5 Q16478 6/20 0.45
GRIK4 Q16099 5/20 0.37
POLB P06746 1/20 0.36
PGR P06401 1/20 0.36
CYP3A4 P08684 1/20 0.36
AR P10275 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9287290 0.90 CA12 (0.47) CA12CA9PARP1GRIK1GRIA1
SCHEMBL8687379 0.86 GRIA1 (0.49) CA12CA9PARP1GRIK1GRIA1
SCHEMBL8589859 0.85 PARP1 (0.53) CA12CA9PARP1GRIK1GRIA1
SCHEMBL8589622 0.84 GRIA1 (0.45) CA12CA9PARP1GRIK1GRIA1
SCHEMBL8688995 0.83 GRIK3 (0.56) CA12CA9PARP1GRIK1GRIA1
SCHEMBL8591048 0.82 GRIA2 (0.47) PARP1GRIK1GRIA1GRIA2GRIA3
SCHEMBL8593265 0.79 CA12 (0.48) CA12CA9PARP1GRIK1GRIA1
SCHEMBL8687373 0.79 CA12 (0.48) CA12CA9PARP1GRIK1GRIA1
SCHEMBL8687221 0.78 GRIA2 (0.59) CA12CA9PARP1GRIK1GRIA1
SCHEMBL8687475 0.77 GRIK3 (0.51) CA12CA9PARP1GRIK1GRIA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0873321-A1 NOVEL AMIDO QUINOXALINE DIONES, THEIR PRODUCTION AND USE BASF AKTIENGESELLSCHAFT (DE) 1998-10-28 EP disclosed