SCHEMBL8594648

SCHEMBL8594648

CC(C)(C)C(=O)N1CCCC(c2ccc(Cl)c(Cl)c2)C1CCN1CCC(O)(c2ccccc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.42
TACR2 P21452 2/20 0.42
RIPK1 Q13546 1/20 0.42
UTS2R Q9UKP6 10/20 0.42
OPRK1 P41145 5/20 0.41
CYP3A4 P08684 4/20 0.41
CYP2D6 P10635 4/20 0.41
ADRA2A P08913 2/20 0.40
ADRA1A P35348 2/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1B P35368 1/20 0.40
MEN1 O00255 1/20 0.40
CES2 O00748 1/20 0.40
SLC22A1 O15245 1/20 0.40
USP2 O75604 1/20 0.40
ABCB11 O95342 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8589466 0.88 TACR1 (0.46) TACR1TACR2UTS2ROPRK1CYP3A4
SCHEMBL8589979 0.84 UTS2R (0.45) TACR1RIPK1UTS2ROPRK1CYP3A4
SCHEMBL8594647 0.82 RIPK1 (0.41) TACR1TACR2RIPK1UTS2ROPRK1
Hydrochloric Acid SCHEMBL8592856 0.77 POLB (0.49) TACR1TACR2DRD2SLC6A2SLC6A4
SCHEMBL8592988 0.76 TACR1 (0.41) TACR1TACR2DRD2DRD4OPRM1
Hydrochloric Acid SCHEMBL8592439 0.75 TACR2 (0.42) TACR1TACR2MEN1LMNADRD2
SCHEMBL8592989 0.73 TACR2 (0.48) TACR1TACR2DRD2DRD1DRD4
Hydrochloric Acid SCHEMBL8593239 0.73 TACR2 (0.49) TACR1TACR2UTS2RCYP3A4CYP2D6
SCHEMBL8589463 0.72 TACR1 (0.42) TACR1TACR2OPRK1OPRM1OPRD1
Hydrochloric Acid SCHEMBL8593273 0.71 UTS2R (0.56) UTS2ROPRK1CYP3A4CYP2D6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5770735-A Polycyclic amine compounds and their enantiomers, their method of preparation and pharmaceutical compositions in which they are present ELF SANOFI (FR) 1998-06-23 US disclosed