SCHEMBL8596332

SCHEMBL8596332

CCOC(=O)c1ccc(CON)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.65
CA2 P00918 4/20 0.65
CA12 O43570 3/20 0.65
CA7 P43166 3/20 0.65
CA9 Q16790 3/20 0.65
CA14 Q9ULX7 3/20 0.65
ESR1 P03372 1/20 0.65
ESR2 Q92731 1/20 0.65
LMNA P02545 1/20 0.62
CYP1A2 P05177 1/20 0.62
CYP3A4 P08684 1/20 0.62
MAOA P21397 1/20 0.62
HTT P42858 3/20 0.57
SMN1; SMN2 Q16637 2/20 0.55
KMT2A Q03164 3/20 0.55
MEN1 O00255 2/20 0.55
STS P08842 1/20 0.53
MAPT P10636 2/20 0.52
AGXT P21549 2/20 0.52
HPGD P15428 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10821032 0.85 CA1 (0.69) CA1CA2CA12CA7CA9
SCHEMBL7746905 0.84 CA1 (0.79) CA1CA2CA12CA7CA9
SCHEMBL10287538 0.84 CA12 (0.67) CA1CA2CA12CA7CA9
SCHEMBL14281812 0.84 CA12 (0.67) CA1CA2CA12CA7CA9
SCHEMBL12935737 0.83 TSHR (0.69) ESR1LMNACYP1A2CYP3A4SMN1; SMN2
SCHEMBL128190 0.83 CA1 (0.70) CA1CA2CA12CA7CA9
SCHEMBL87450 0.82 CA1 (0.83) CA1CA2CA12CA7CA9
SCHEMBL6665051 0.82 CA12 (0.65) CA1CA2CA12CA7CA9
SCHEMBL1520636 0.81 LOXL2 (0.67) CA1CA2CA12CA7CA9
SCHEMBL687664 0.81 LOXL2 (0.67) CA1CA2CA12CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726314-A ACETYLCHOLINESTERASE INHIBITORS AS NERVE AGENT ANTIDOTES GEORGIA TECH RESEARCH CORP. (US) 1998-03-10 US disclosed
US-5714615-A ACETYLCHOLINESTERASE ENZYME INHIBITOR, STIMULATE NICOTINIC RECEPTORS IN CENTRAL NERVOUS SYSTEM GEORGIA TECH RESEARCH CORPORATION (US) 1998-02-03 US disclosed
WO-1995021822-A1 PYRIDINIUM COMPOUNDS GEORGIA TECH RESEARCH CORPORATION (US) 1995-08-17 WO disclosed
US-5290942-A Acetylcholinesterase inhibitors GEORGIA TECH RESEARCH CORPORATION (US) 1994-03-01 US disclosed
US-5206371-A Acetylcholinesterase inhibitor GEORGIA TECH RESEARCH CORPORATION (US) 1993-04-27 US disclosed
US-5180831-A Acetylcholinesterase Inhibitors GEORGIA TECH RESEARCH CORPORATION (US) 1993-01-19 US disclosed
EP-0361067-B1 DISUBSTITUTED NAPHTHALINES, PREPARATION PROCESSES AND THEIR HERBICIDAL USE BAYER AG (DE) 1992-11-11 EP disclosed
US-5108489-A HERBICIDAL DISUBSTITUTED NAPHTHALENES BAYER AKTIENGESELLSCHAFT (DE) 1992-04-28 US disclosed
EP-0470430-A1 Process for the preparation of oxyguanidins BAYER AG (DE) 1992-02-12 EP disclosed
US-5086177-A Chemical intermediate for herbicides BAYER AKTIENGESELLSCHAFT (DE) 1992-02-04 US disclosed
US-4980469-A Reacting isothiourea of nitrogen containing heterocycle with hydroxylamine derivative BAYER AKTIENGESELLSCHAFT (DE) 1990-12-25 US disclosed
EP-0361067-A1 Disubstituted naphthalines, preparation processes and their herbicidal use BAYER AG (DE) 1990-04-04 EP disclosed
EP-0358018-A2 Process for the preparation of oxyguanidines BAYER AG (DE) 1990-03-14 EP disclosed
US-4725304-A HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1988-02-16 US disclosed
EP-0224078-A1 Thienyl sulfonyl guanidine derivatives BAYER AG (DE) 1987-06-03 EP disclosed
EP-0173956-A1 Sulfonyl-guanidinotriazine derivatives BAYER AG (DE) 1986-03-12 EP disclosed
EP-0173317-A1 Unsymmetrical sulfonyl guanidines BAYER AG (DE) 1986-03-05 EP disclosed