SCHEMBL8598652

SCHEMBL8598652

O=[N+]([O-])c1ccc(CSP(=O)(O)O)c([N+](=O)[O-])c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.55
ALOX5 P09917 1/20 0.48
ALDH1A1 P00352 5/20 0.47
GPR35 Q9HC97 2/20 0.47
TP53 P04637 1/20 0.47
HPGD P15428 1/20 0.47
TSHR P16473 1/20 0.47
MAPK1 P28482 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
TXNRD1 Q16881 1/20 0.46
TXNRD3 Q86VQ6 1/20 0.46
TXNRD2 Q9NNW7 1/20 0.46
TDP1 Q9NUW8 2/20 0.45
HIF1A Q16665 1/20 0.44
MAPT P10636 4/20 0.43
GAA P10253 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8598555 0.80 CYP1A2 (0.60) CYP1A2ALOX5ALDH1A1GPR35TP53
SCHEMBL12727872 0.78 CYP1A2 (0.57) CYP1A2ALOX5ALDH1A1GPR35TP53
SCHEMBL27543660 0.78 CYP1A2 (0.57) CYP1A2ALOX5ALDH1A1GPR35TP53
SCHEMBL1742521 0.78 CYP1A2 (0.57) CYP1A2ALOX5ALDH1A1GPR35TP53
SCHEMBL27961047 0.76 CYP1A2 (0.68) CYP1A2ALOX5ALDH1A1GPR35TP53
SCHEMBL8599963 0.76 CYP1A2 (0.59) CYP1A2ALOX5ALDH1A1GPR35TP53
SCHEMBL28738722 0.76 CYP1A2 (0.55) CYP1A2ALOX5ALDH1A1GPR35TP53
SCHEMBL8600350 0.76 IDO1 (0.56) CYP1A2ALDH1A1TSHRMAPTAKR1C3
SCHEMBL3124261 0.75 CYP1A2 (0.67) CYP1A2ALOX5ALDH1A1GPR35TP53
SCHEMBL3776333 0.75 IDO1 (0.63) CYP1A2ALOX5ALDH1A1GPR35TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0723973-B1 Nucleoside phosphorothioate derivatives, synthesis and use thereof KING S COLLEGE LONDON (GB) 1998-10-21 EP disclosed
US-5708161-A Nucleoside phosphorothioate derivatives, synthesis and use thereof KING'S COLLEGE LONDON (GB) 1998-01-13 US disclosed
EP-0723973-A1 Nucleoside phosphorothioate derivatives, synthesis and use thereof KING'S COLLEGE LONDON (GB) 1996-07-31 EP disclosed