SCHEMBL8600350

SCHEMBL8600350

O=[N+]([O-])c1ccc(CSP(=O)(O)O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.56
AKR1C3 P42330 1/20 0.56
CYP2C19 P33261 3/20 0.53
CYP1A2 P05177 2/20 0.53
CYP2C9 P11712 1/20 0.53
TSHR P16473 1/20 0.50
LOXL2 Q9Y4K0 1/20 0.48
ALDH1A1 P00352 2/20 0.47
CA1 P00915 2/20 0.47
CA2 P00918 1/20 0.47
CES2 O00748 1/20 0.47
CES1 P23141 1/20 0.47
MAPT P10636 2/20 0.45
BCHE P06276 1/20 0.45
ACHE P22303 1/20 0.45
GFER P55789 1/20 0.44
LMNA P02545 1/20 0.44
CA12 O43570 1/20 0.44
MMP2 P08253 1/20 0.44
MMP9 P14780 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3244320 0.77 CYP2C19 (0.63) IDO1CYP2C19CYP1A2CYP2C9TSHR
SCHEMBL1035377 0.77 CYP2C19 (0.81) IDO1CYP2C19CYP1A2CYP2C9TSHR
Phosphoric Acid SCHEMBL28639141 0.76 CA1 (0.65) AKR1C3TSHRALDH1A1CA1CA2
SCHEMBL8598652 0.76 CYP1A2 (0.55) AKR1C3CYP1A2TSHRALDH1A1MAPT
SCHEMBL11040755 0.76 AKR1C3 (0.61) IDO1AKR1C3CYP2C19CYP1A2TSHR
SCHEMBL916699 0.76 AKR1C3 (0.61) IDO1AKR1C3CYP2C19CYP1A2TSHR
Paranitrobenzyl Alcohol SCHEMBL28005884 0.76 AKR1C3 (0.61) IDO1AKR1C3CYP2C19CYP1A2CYP2C9
SCHEMBL7244787 0.75 CYP2C19 (0.79) IDO1CYP2C19CYP1A2CYP2C9TSHR
SCHEMBL8648393 0.74 AKR1C3 (0.59) IDO1AKR1C3CYP2C19CYP1A2CYP2C9
SCHEMBL8600352 0.74 IDO1 (0.39) IDO1AKR1C3CYP2C19CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0723973-B1 Nucleoside phosphorothioate derivatives, synthesis and use thereof KING S COLLEGE LONDON (GB) 1998-10-21 EP disclosed
US-5708161-A Nucleoside phosphorothioate derivatives, synthesis and use thereof KING'S COLLEGE LONDON (GB) 1998-01-13 US disclosed
EP-0723973-A1 Nucleoside phosphorothioate derivatives, synthesis and use thereof KING'S COLLEGE LONDON (GB) 1996-07-31 EP disclosed