SCHEMBL8599203

SCHEMBL8599203

COC(=O)CSc1cc(N)c(F)cc1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
MAPT P10636 4/20 0.43
HSD17B10 Q99714 3/20 0.43
HPGD P15428 3/20 0.43
TP53 P04637 1/20 0.43
KMT2A Q03164 4/20 0.42
POLB P06746 2/20 0.42
RXFP1 Q9HBX9 2/20 0.42
PRNP P04156 1/20 0.42
GAA P10253 3/20 0.41
GLA P06280 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MEN1 O00255 2/20 0.38
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
GFER P55789 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8603065 0.86 KDM4E (0.48) ALDH1A1MAPTHSD17B10HPGDTP53
SCHEMBL8599957 0.85 CCNB2 (0.35) ALDH1A1MAPTKMT2APOLBRXFP1
SCHEMBL8598571 0.85 ALDH1A1 (0.42) ALDH1A1MAPTHSD17B10HPGDKMT2A
SCHEMBL8603159 0.84 ALDH1A1 (0.42) ALDH1A1HSD17B10HPGDTP53POLB
SCHEMBL8601923 0.82 FABP4 (0.40) ALDH1A1RXFP1PRNPKDM4ECYP1A2
SCHEMBL8599557 0.82 ALDH1A1 (0.43) ALDH1A1MAPTHSD17B10HPGDKMT2A
SCHEMBL8603934 0.82 MAPT (0.33) ALDH1A1MAPTHSD17B10HPGDKMT2A
SCHEMBL8602507 0.81 TDP1 (0.34) ALDH1A1MAPTHSD17B10HPGDKMT2A
SCHEMBL8603132 0.81 ALDH1A1 (0.41) ALDH1A1MAPTHSD17B10KMT2APOLB
SCHEMBL8598803 0.79 ALDH1A1 (0.39) ALDH1A1MAPTHSD17B10HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626370-B1 Process for producing aromatic isothiocyanate derivatives SUMITOMO CHEMICAL CO (JP) 1998-02-11 EP disclosed
US-5631209-A ALGICIDES ROHM AND HAAS COMPANY (US) 1997-05-20 US disclosed
EP-0523244-B1 SALT OF DITHIOCARBAMIC ACID, PRODUCTION THEREOF, AND PRODUCTION OF ISOTHIOCYANATE FROM SAID SALT IHARA CHEMICAL IND CO (JP) 1996-04-10 EP disclosed
EP-0415642-B1 Glutarimides ROHM & HAAS (US) 1995-12-06 EP disclosed
US-5393735-A N-(halo-oxy-)phenyl substituted cyclic imides ROHM AND HAAS COMPANY (US) 1995-02-28 US disclosed
EP-0626370-A1 Process for producing aromatic isothiocyanate derivatives SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1994-11-30 EP disclosed
EP-0415641-B1 Substituted glutaramic acids and derivatives ROHM & HAAS (US) 1994-01-19 EP disclosed
US-5274166-A Dithiocarbamic acid salt, process for production thereof, and process for production of isothiocyanate using said dithiocarbamic acid salt IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 1993-12-28 US disclosed
US-5238908-A HERBICIDAL GLUTARAMIC ACIDS AND DERIVATIVES ROHM AND HAAS COMPANY (US) 1993-08-24 US disclosed
EP-0523244-A1 SALT OF DITHIOCARBAMIC ACID, PRODUCTION THEREOF, AND PRODUCTION OF ISOTHIOCYANATE FROM SAID SALT IHARA CHEMICAL INDUSTRY Co., Ltd. (JP) 1993-01-20 EP disclosed
EP-0415641-A1 Substituted glutaramic acids and derivatives ROHM AND HAAS COMPANY (US) 1991-03-06 EP disclosed
EP-0415642-A1 Glutarimides ROHM AND HAAS COMPANY (US) 1991-03-06 EP disclosed