SCHEMBL8599424

SCHEMBL8599424

C=C(C)c1cc2ccc(OC)cc2s1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.49
DYRK1A Q13627 4/20 0.46
CLK1 P49759 4/20 0.46
DYRK1B Q9Y463 1/20 0.46
CHRNA7 P36544 3/20 0.44
CYP1A2 P05177 3/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2C19 P33261 2/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
HTT P42858 1/20 0.44
HDAC1 Q13547 2/20 0.41
PDGFRB P09619 1/20 0.41
PDGFRA P16234 1/20 0.41
PDK1 Q15118 1/20 0.41
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
TUBA1B P68363 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9623048 0.87 CLK1 (0.60) CA2DYRK1ACLK1DYRK1BBACE1
SCHEMBL914782 0.80 BCL2L1 (0.54) CA2DYRK1ACLK1DYRK1BCHRNA7
SCHEMBL13709512 0.79 F9 (0.56) CA2DYRK1ACLK1DYRK1BCHRNA7
SCHEMBL31207841 0.79 HDAC1 (0.56) CA2DYRK1ACLK1DYRK1BCHRNA7
SCHEMBL29020102 0.79 BCL2L1 (0.53) CA2DYRK1ACLK1DYRK1BCHRNA7
SCHEMBL1098993 0.79 HDAC1 (0.56) CA2DYRK1ACLK1DYRK1BCHRNA7
SCHEMBL30298109 0.78 CLK1 (0.48) CA2DYRK1ACLK1DYRK1BCHRNA7
Potassium Ion SCHEMBL25233840 0.78 CLK1 (0.50) CA2DYRK1ACLK1DYRK1BCHRNA7
SCHEMBL22590860 0.77 HDAC1 (0.60) DYRK1ACLK1DYRK1BCHRNA7CYP1A2
SCHEMBL5542989 0.75 CA2 (0.54) CA2DYRK1ACYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641791-B1 NOVEL BENZOTHIOPHENE DERIVATIVE TEIKOKU HORMONE MFG CO LTD (JP) 1998-01-28 EP disclosed
US-5472962-A Antiestrogenic agents TEIKOKU HORMONE MFG. CO., LTD. (JP) 1995-12-05 US disclosed
EP-0641791-A1 NOVEL BENZOTHIOPHENE DERIVATIVE TEIKOKU HORMONE MFG. CO., LTD. (JP) 1995-03-08 EP disclosed