SCHEMBL8599586

SCHEMBL8599586

COc1ccc2cc(C3=CCCC3)sc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
CA2 P00918 1/20 0.43
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C19 P33261 1/20 0.37
ACHE P22303 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
TP53 P04637 1/20 0.36
PDK1 Q15118 1/20 0.36
BACE1 P56817 1/20 0.36
CYP2A6 P11509 1/20 0.35
PSMB8 P28062 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
PDGFRB P09619 1/20 0.35
PDGFRA P16234 1/20 0.35
CDK1 P06493 1/20 0.34
MAPKAPK2 P49137 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6836981 0.96 NPC1 (0.53) NPC1RAB9ACA2CYP1A2CYP3A4
SCHEMBL8601704 0.94 NPC1 (0.52) NPC1RAB9ACA2CYP1A2CYP3A4
SCHEMBL8599883 0.94 NPC1 (0.52) NPC1RAB9ACA2CYP1A2CYP3A4
SCHEMBL8600780 0.94 NPC1 (0.52) NPC1RAB9ACA2CYP1A2CYP3A4
SCHEMBL8600782 0.94 NPC1 (0.52) NPC1RAB9ACA2CYP1A2CYP3A4
SCHEMBL8601702 0.94 NPC1 (0.52) NPC1RAB9ACA2CYP1A2CYP3A4
SCHEMBL8601706 0.94 NPC1 (0.52) NPC1RAB9ACA2CYP1A2CYP3A4
SCHEMBL8596151 0.80 CA2 (0.44) NPC1RAB9ACA2CYP1A2CYP3A4
SCHEMBL6312469 0.80 HTR6 (0.49) CA2CYP1A2CYP3A4MEN1MAPK1
SCHEMBL8599155 0.79 CA2 (0.40) NPC1RAB9ACA2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641791-B1 NOVEL BENZOTHIOPHENE DERIVATIVE TEIKOKU HORMONE MFG CO LTD (JP) 1998-01-28 EP disclosed
US-5472962-A Antiestrogenic agents TEIKOKU HORMONE MFG. CO., LTD. (JP) 1995-12-05 US disclosed
EP-0641791-A1 NOVEL BENZOTHIOPHENE DERIVATIVE TEIKOKU HORMONE MFG. CO., LTD. (JP) 1995-03-08 EP disclosed