SCHEMBL8600000

SCHEMBL8600000

O=C(O)C1CC(=O)N1CO

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 4/20 0.37
ITGA5 P08648 4/20 0.37
SIGMAR1 Q99720 1/20 0.35
ACE P12821 4/20 0.34
ITGB3 P05106 2/20 0.34
ITGAV P06756 2/20 0.34
ITGA4 P13612 2/20 0.34
POLB P06746 3/20 0.33
MME P08473 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MAPT P10636 1/20 0.33
BRD4 O60885 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8866460 0.83 BRD4 (0.35) ITGB1ITGA5ACEITGB3ITGAV
SCHEMBL29954394 0.81 ITGB1 (0.39) ITGB1ITGA5ACEITGB3ITGAV
SCHEMBL21424968 0.81 ITGB1 (0.39) ITGB1ITGA5ACEITGB3ITGAV
SCHEMBL7403414 0.76 ITGB1 (0.33) ITGB1ITGA5ACEITGB3ITGAV
SCHEMBL2535132 0.74 EHMT2 (0.47) ITGB1ITGA5ACEGAA
SCHEMBL10345901 0.74 ACE (0.33) ITGB1ITGA5ACEITGB3ITGAV
SCHEMBL10345950 0.74 ACE (0.33) ITGB1ITGA5ACEITGB3ITGAV
SCHEMBL2535135 0.74 EHMT2 (0.47) ITGB1ITGA5ACEGAA
SCHEMBL7406627 0.73 ITGB1 (0.41) ITGB1ITGA5ITGB3ITGAVITGA4
SCHEMBL29127664 0.70 SIGMAR1 (0.42) SIGMAR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998612-A Antibiotic synthesis MERCK SHARP & DOHME CORP. 1999-12-07 US disclosed
EP-0171159-B1 SUBSTITUTED AZETIDINONE COMPOUNDS, THEIR PREPARATION, AND MEDICAMENTS CONTAINING THEM YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1990-05-30 EP disclosed
EP-0078026-B1 ANTIBIOTIC SYNTHESIS MERCK & CO. INC. (US) 1988-09-28 EP disclosed
US-4719207-A CENTRAL NERVOUS SYSTEM YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1988-01-12 US disclosed
EP-0171159-A1 Substituted azetidinone compounds, their preparation, and medicaments containing them YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1986-02-12 EP disclosed
EP-0078026-A2 Antibiotic synthesis MERCK & CO. INC. (US) 1983-05-04 EP disclosed