SCHEMBL8600352

SCHEMBL8600352

O=[N+](O)c1ccc(CSP(=O)([O-])O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.39
AKR1C3 P42330 1/20 0.39
CYP2C19 P33261 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.33
MAPT P10636 3/20 0.32
BCHE P06276 1/20 0.32
ACHE P22303 1/20 0.32
ALDH1A1 P00352 4/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
LOXL2 Q9Y4K0 1/20 0.32
LMNA P02545 3/20 0.31
HTT P42858 2/20 0.31
THRB P10828 1/20 0.31
HPGD P15428 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2374254 0.77 AKR1C3 (0.42) IDO1AKR1C3CYP2C19CYP1A2TSHR
SCHEMBL8600350 0.74 IDO1 (0.56) IDO1AKR1C3CYP2C19CYP1A2CYP2C9
SCHEMBL3625606 0.74 TSHR (0.42) AKR1C3CYP2C19TSHRMAPTALDH1A1
SCHEMBL5983777 0.72 AKR1C3 (0.58) IDO1AKR1C3TSHRMAPTALDH1A1
Phosphonic Acid SCHEMBL5328144 0.72 TSHR (0.38) IDO1AKR1C3TSHRMAPTALDH1A1
SCHEMBL735220 0.70 AKR1C3 (0.44) IDO1AKR1C3TSHRMAPTALDH1A1
SCHEMBL356641 0.70 CA2 (0.37) AKR1C3TSHRCA1CA2CES2
SCHEMBL8133189 0.69 GSK3B (0.42) AKR1C3TSHRMAPTALDH1A1CA1
SCHEMBL8601137 0.68 AKR1C3 (0.53) IDO1AKR1C3TSHRALDH1A1CA1
SCHEMBL5002727 0.67 TSHR (0.41) IDO1AKR1C3CYP2C19CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0723973-B1 Nucleoside phosphorothioate derivatives, synthesis and use thereof KING S COLLEGE LONDON (GB) 1998-10-21 EP disclosed
US-5708161-A Nucleoside phosphorothioate derivatives, synthesis and use thereof KING'S COLLEGE LONDON (GB) 1998-01-13 US disclosed
EP-0723973-A1 Nucleoside phosphorothioate derivatives, synthesis and use thereof KING'S COLLEGE LONDON (GB) 1996-07-31 EP disclosed