SCHEMBL8600596

SCHEMBL8600596

CCCC(CCC)=C(C#N)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 4/20 0.40
HDAC1 Q13547 4/20 0.40
HDAC2 Q92769 4/20 0.40
HDAC8 Q9BY41 4/20 0.40
FFAR3 O14843 3/20 0.40
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
TSHR P16473 5/20 0.33
ALDH1A1 P00352 4/20 0.32
KMT2A Q03164 2/20 0.31
MAPT P10636 1/20 0.31
AKR1B1 P15121 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
LMNA P02545 1/20 0.31
MAPK1 P28482 1/20 0.31
PPARG P37231 6/20 0.30
PPARD Q03181 6/20 0.30
PPARA Q07869 6/20 0.30
HDAC11 Q96DB2 5/20 0.30
GPR84 Q9NQS5 4/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7552128 0.92 CES1 (0.39) HDAC3HDAC1HDAC2HDAC8FFAR3
SCHEMBL3923583 0.91 FFAR3 (0.37) HDAC3HDAC1HDAC2HDAC8FFAR3
SCHEMBL19357539 0.91 FFAR3 (0.37) HDAC3HDAC1HDAC2HDAC8FFAR3
SCHEMBL7546476 0.87 CES1 (0.41) CES2CES1TSHRALDH1A1KMT2A
SCHEMBL1074448 0.85 AKR1B1 (0.46) CES2CES1TSHRALDH1A1KMT2A
SCHEMBL7544283 0.85 FFAR3 (0.32) HDAC3HDAC1HDAC2HDAC8FFAR3
SCHEMBL7542632 0.84 AKR1B1 (0.45) CES2CES1TSHRALDH1A1KMT2A
SCHEMBL31625063 0.84 KMT2A (0.48) CES2CES1TSHRALDH1A1KMT2A
SCHEMBL11910004 0.84 KMT2A (0.48) CES2CES1TSHRALDH1A1KMT2A
SCHEMBL7542466 0.82 KMT2A (0.47) CES2CES1TSHRALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5734061-A Process for preparing spirocyclic lactams SMITHKLINE BEECHAM CORPORATION (US) 1998-03-31 US disclosed