SCHEMBL3923583

SCHEMBL3923583

CCCC(CC)=C(C#N)C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FFAR3 O14843 4/20 0.37
HDAC3 O15379 3/20 0.37
HDAC1 Q13547 3/20 0.37
HDAC2 Q92769 3/20 0.37
HDAC8 Q9BY41 3/20 0.37
ALDH1A1 P00352 1/20 0.34
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19357539 1.00 FFAR3 (0.37) FFAR3HDAC3HDAC1HDAC2HDAC8
SCHEMBL8600596 0.91 HDAC3 (0.40) FFAR3HDAC3HDAC1HDAC2HDAC8
SCHEMBL7545293 0.88 CES1 (0.39) ALDH1A1CES2CES1TSHR
SCHEMBL188481 0.87 FFAR3 (0.36) FFAR3ALDH1A1TSHR
SCHEMBL8673175 0.86 AKR1B1 (0.43) ALDH1A1CES2CES1TSHR
SCHEMBL8673179 0.86 AKR1B1 (0.43) ALDH1A1CES2CES1TSHR
SCHEMBL540776 0.85 GPR84 (0.45) ALDH1A1CES2CES1TSHR
SCHEMBL7552128 0.84 CES1 (0.39) FFAR3HDAC3HDAC1HDAC2HDAC8
SCHEMBL23204219 0.82 MAPK10 (0.39) FFAR3HDAC3HDAC1HDAC2HDAC8
SCHEMBL23163159 0.82 MAPK10 (0.39) FFAR3HDAC3HDAC1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017158151-A1 PYRIMIDONE DERIVATIVES AND THEIR USE IN THE TREATMENT, AMELIORATION OR PREVENTION OF A VIRAL DISEASE SAVIRA PHARMACEUTICALS GMBH (AT) 2017-09-21 WO disclosed
EP-1807457-A4 VINYL CHLORIDE RESIN COMPOSITION AND METHOD FOR PREPARATION THEREOF LG CHEMICAL LTD (KR) 2009-03-25 EP disclosed
EP-1807457-A1 VINYL CHLORIDE RESIN COMPOSITION AND METHOD FOR PREPARATION THEREOF LG Chem, Ltd. (KR) 2007-07-18 EP disclosed
WO-2006049392-A1 VINYL CHLORIDE RESIN COMPOSITION AND METHOD FOR PREPARATION THEREOF LG CHEM, LTD. (KR) 2006-05-11 WO disclosed
US-5843951-A Analgesic composition of pyrazolo(1,5-A) pyrimidines OTSUKA PHARMACEUTICAL FACTORY INC. (JP) 1998-12-01 US disclosed
EP-0795555-A1 ANALGESICS OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1997-09-17 EP disclosed