SCHEMBL8600869

SCHEMBL8600869

CS(=O)(=O)Oc1ccc2c(c1)C(=O)CC2

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.48
CA5A P35218 1/20 0.48
PBRM1 Q86U86 1/20 0.47
HRH3 Q9Y5N1 2/20 0.47
BRD4 O60885 3/20 0.46
ALDH1A1 P00352 2/20 0.44
MAOB P27338 5/20 0.43
MAOA P21397 3/20 0.43
PTGS2 P35354 2/20 0.42
HPGD P15428 1/20 0.41
STS P08842 1/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14128769 0.90 MAOA (0.53) CA2CA5AHRH3ALDH1A1MAOB
SCHEMBL5685785 0.88 MAOB (0.49) CA2CA5AHRH3ALDH1A1MAOB
SCHEMBL1513396 0.81 MAOB (0.46) CA2PBRM1HRH3BRD4MAOB
SCHEMBL251842 0.79 MAOB (0.54) PBRM1HRH3BRD4ALDH1A1MAOB
SCHEMBL29392039 0.79 MAOB (0.54) PBRM1HRH3BRD4ALDH1A1MAOB
SCHEMBL3821515 0.79 MAOB (0.55) MAOBMAOA
SCHEMBL6130607 0.77 MAPK14 (0.56) MAOBKDM4E
SCHEMBL30103244 0.75 HRH3 (0.56) PBRM1HRH3BRD4MAOBMAOA
SCHEMBL29308778 0.75 STS (0.62) CA2CA5AALDH1A1HPGDSTS
SCHEMBL6184702 0.75 STS (0.68) CA2CA5AHRH3ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0657426-B1 Tricyclic pyrrole derivatives HOFFMANN LA ROCHE (CH) 1998-07-22 EP disclosed
US-5646173-A ANTISEROTONINE AGENTS; CENTRAL NERVOUS SYSTEM DISORDERS; ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1997-07-08 US disclosed
EP-0657426-A2 Tricyclic pyrrole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1995-06-14 EP disclosed