SCHEMBL8600959

SCHEMBL8600959

O=CCC1Cc2ccc(Br)cc2C1=O

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
METAP1 P53582 10/20 0.50
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PARP1 P09874 1/20 0.37
PARP10 Q53GL7 1/20 0.37
S100A4 P26447 1/20 0.35
ACHE P22303 2/20 0.35
PBRM1 Q86U86 1/20 0.35
TDP2 O95551 1/20 0.34
CYP19A1 P11511 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8874550 1.00 METAP1 (0.50) METAP1TDP1L3MBTL1PARP1PARP10
SCHEMBL8600862 0.84 METAP1 (0.47) METAP1TDP1L3MBTL1PARP1PARP10
SCHEMBL8874447 0.84 METAP1 (0.47) METAP1TDP1L3MBTL1PARP1PARP10
SCHEMBL8600861 0.84 METAP1 (0.47) METAP1TDP1L3MBTL1PARP1PARP10
SCHEMBL8873164 0.81 METAP1 (0.50) METAP1PARP1PARP10S100A4ACHE
SCHEMBL8598468 0.81 METAP1 (0.50) METAP1PARP1PARP10S100A4ACHE
SCHEMBL8598137 0.81 METAP1 (0.67) METAP1PARP1PARP10ACHE
SCHEMBL8873958 0.81 ACHE (0.55) METAP1PARP1PARP10ACHE
SCHEMBL8875167 0.81 METAP1 (0.67) METAP1PARP1PARP10ACHE
SCHEMBL8594761 0.81 ACHE (0.55) METAP1PARP1PARP10ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0657426-B1 Tricyclic pyrrole derivatives HOFFMANN LA ROCHE (CH) 1998-07-22 EP disclosed
US-5646173-A ANTISEROTONINE AGENTS; CENTRAL NERVOUS SYSTEM DISORDERS; ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1997-07-08 US disclosed
EP-0657426-A2 Tricyclic pyrrole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1995-06-14 EP disclosed