SCHEMBL8601161

SCHEMBL8601161

CONC(=O)Cn1c(C(F)(F)F)nc2c(NC(=O)c3c(Cl)cccc3Cl)cccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.46
PTGES O14684 6/20 0.41
MMP2 P08253 1/20 0.39
BRD4 O60885 1/20 0.38
CREBBP Q92793 1/20 0.38
HTT P42858 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
TYK2 P29597 1/20 0.37
POLB P06746 1/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
ALDH1A1 P00352 1/20 0.36
APEX1 P27695 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8602410 0.89 TP53 (0.45) TP53PTGESMMP2HTTMEN1
SCHEMBL8596165 0.87 TP53 (0.45) TP53PTGESMMP2HTTMEN1
SCHEMBL8597372 0.86 PTGES (0.45) TP53PTGESBRD4CREBBPMEN1
SCHEMBL8597312 0.86 TP53 (0.43) TP53PTGESMMP2HTTMEN1
SCHEMBL8596007 0.86 TP53 (0.51) TP53HTTMEN1KMT2AL3MBTL1
SCHEMBL8596981 0.86 TP53 (0.44) TP53PTGESMMP2HTTMEN1
SCHEMBL8602225 0.85 TP53 (0.44) TP53PTGESMMP2HTTMEN1
SCHEMBL8600307 0.85 TP53 (0.44) TP53PTGESMMP2HTTSMN1; SMN2
SCHEMBL8597745 0.85 S1PR2 (0.47) TP53HTTMEN1KMT2ASMN1; SMN2
SCHEMBL8595161 0.85 PTGES (0.42) TP53PTGESTYK2LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863881-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE IN THE PREVENTION AND/OR THE TREATMENT OF BONE DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-09-16 EP disclosed
WO-1997010219-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE IN THE PREVENTION AND/OR THE TREATMENT OF BONE DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-03-20 WO disclosed