SCHEMBL8601768

SCHEMBL8601768

C=CCc1cc(-c2ccccn2)ccc1C#CCCCC(C)F

nearest known ligand 0.32

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP19A1 P11511 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
SQOR Q9Y6N5 1/20 0.32
OPRD1 P41143 2/20 0.31
CCNE1 P24864 1/20 0.31
CDK2 P24941 1/20 0.31
PDK2 Q15119 1/20 0.31
ADRA2A P08913 1/20 0.30
ADRA2B P18089 1/20 0.30
ADRA2C P18825 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8599902 0.89
SCHEMBL8603951 0.87 SQOR (0.33) SQORCCNE1CDK2PDK2
SCHEMBL8601985 0.84 SQOR (0.38) CYP1A2CYP2D6CYP19A1CYP2C9CYP2C19
SCHEMBL8601802 0.83 GABRA1 (0.31)
SCHEMBL8601487 0.83 SQOR (0.32) SQOR
SCHEMBL8601987 0.81 SQOR (0.40) CYP1A2CYP2D6CYP19A1CYP2C9CYP2C19
SCHEMBL8600854 0.79 CYP1A2 (0.34) CYP1A2CYP2D6CYP19A1CYP2C9CYP2C19
SCHEMBL8600713 0.77 PIK3CD (0.34) CYP1A2CYP2D6CYP19A1CYP2C9CYP2C19
SCHEMBL8601776 0.75 PTAFR (0.31)
SCHEMBL8598141 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5779934-A FLUORINATING AN ALCOHOL DERIVATIVE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-07-14 US disclosed