SCHEMBL8604142

SCHEMBL8604142

O=C(OCc1ccccc1)OC(=O)[C@@H]1C[C@@H](O)CN1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
TSHR P16473 1/20 0.41
HTR2C P28335 1/20 0.41
CTSC P53634 1/20 0.40
BACE1 P56817 1/20 0.39
GLA P06280 1/20 0.39
MAPK1 P28482 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A3 Q01959 1/20 0.39
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
GAA P10253 1/20 0.39
FABP7 O15540 1/20 0.38
FABP5 Q01469 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8602762 1.00 ALDH1A1 (0.43) ALDH1A1TSHRHTR2CCTSCBACE1
SCHEMBL1077276 0.89 TSHR (0.51) ALDH1A1TSHRHTR2CCTSCBACE1
SCHEMBL7382311 0.89 TSHR (0.51) ALDH1A1TSHRHTR2CCTSCBACE1
SCHEMBL10137745 0.89 TSHR (0.51) ALDH1A1TSHRHTR2CCTSCBACE1
SCHEMBL9636938 0.89 TSHR (0.51) ALDH1A1TSHRHTR2CCTSCBACE1
SCHEMBL23485377 0.89 TSHR (0.51) ALDH1A1TSHRHTR2CCTSCBACE1
SCHEMBL21961574 0.89 TSHR (0.51) ALDH1A1TSHRHTR2CCTSCBACE1
Hydrochloric Acid SCHEMBL7382305 0.88 TSHR (0.53) ALDH1A1TSHRHTR2CCTSCBACE1
Hydrochloric Acid SCHEMBL1784263 0.88 TSHR (0.53) ALDH1A1TSHRHTR2CCTSCBACE1
SCHEMBL6167045 0.86 CTSC (0.46) ALDH1A1TSHRHTR2CCTSCBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828851-A2 TRIPEPTIDYLPEPTIDASE INHIBITORS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1998-03-18 EP disclosed
WO-1996035805-A2 TRIPEPTIDYLPEPTIDASE INHIBITORS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1996-11-14 WO disclosed