SCHEMBL6167045

SCHEMBL6167045

O=C(OCc1ccccc1)OC(=O)[C@@H]1CC(F)CN1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSC P53634 3/20 0.46
ALDH1A1 P00352 4/20 0.42
TSHR P16473 1/20 0.41
HTR2C P28335 1/20 0.40
BACE1 P56817 1/20 0.38
GLA P06280 1/20 0.38
MAPK1 P28482 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A3 Q01959 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8607040 1.00 CTSC (0.46) CTSCALDH1A1TSHRHTR2CBACE1
SCHEMBL20745388 0.89 CTSC (0.50) CTSCALDH1A1TSHRHTR2CBACE1
SCHEMBL16407831 0.89 CTSC (0.50) CTSCALDH1A1TSHRHTR2CBACE1
SCHEMBL12480861 0.89 CTSC (0.50) CTSCALDH1A1TSHRHTR2CBACE1
SCHEMBL21964312 0.89 CTSC (0.50) CTSCALDH1A1TSHRHTR2CBACE1
SCHEMBL19388654 0.89 CTSC (0.50) CTSCALDH1A1TSHRHTR2CBACE1
Hydrochloric Acid SCHEMBL25201793 0.88 TSHR (0.52) CTSCALDH1A1TSHRHTR2CBACE1
Hydrochloric Acid SCHEMBL29820504 0.88 TSHR (0.52) CTSCALDH1A1TSHRHTR2CBACE1
SCHEMBL8602762 0.86 ALDH1A1 (0.43) CTSCALDH1A1TSHRHTR2CBACE1
SCHEMBL8604142 0.86 ALDH1A1 (0.43) CTSCALDH1A1TSHRHTR2CBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465891-A4 INHIBITORS OF DIPEPTIDYL PEPTIDASE IV GUILFORD PHARM INC (US) 2005-08-17 EP disclosed
EP-1465891-A2 INHIBITORS OF DIPEPTIDYL PEPTIDASE IV GUILFORD PHARMACEUTICALS INC. (US) 2004-10-13 EP disclosed
WO-2003057666-A2 INHIBITORS OF DIPEPTIDYL PEPTIDASE IV GUILFORD PHARMACEUTICALS (US) 2003-07-17 WO disclosed
WO-2003057144-A2 CHANGE INHIBITORS OF DIPEPTIDYL PEPTIDASE IV GUILFORD PHARMACEUTICALS (US) 2003-07-17 WO disclosed