SCHEMBL8604252

SCHEMBL8604252

CS(=O)(=O)c1ccc(-c2ccccc2CCN)cc1

nearest known ligand 0.59

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.59
DRD1 P21728 1/20 0.50
PTGS1 P23219 1/20 0.47
HSD11B1 P28845 1/20 0.46
KIF11 P52732 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8604437 0.85 PTGS2 (0.61) PTGS2DRD1PTGS1
SCHEMBL13675349 0.83 PTGS2 (0.67) PTGS2DRD1PTGS1
SCHEMBL5723494 0.81 PTGS2 (0.65) PTGS2DRD1PTGS1
SCHEMBL9890741 0.78 PTGS2 (0.56) PTGS2DRD1PTGS1
SCHEMBL8487915 0.78 PTGS2 (0.75) PTGS2DRD1PTGS1
SCHEMBL6048541 0.77 PTGS2 (0.59) PTGS2DRD1PTGS1
SCHEMBL9839608 0.77 TAAR1 (0.52)
SCHEMBL1868872 0.77 DPP4 (0.68)
Hydrochloric Acid SCHEMBL6048552 0.76 PTGS2 (0.57) PTGS2DRD1PTGS1
SCHEMBL5502727 0.75 PTGS2 (1.00) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5723489-A ADRENERGIC BLOCKING AGENTS OR STIMULANTS FOR GASTROINTESTINAL DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-03-03 US disclosed