SCHEMBL8604254

SCHEMBL8604254

CS(=O)(=O)c1ccc(C(CN)c2ccccc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.59
TAAR1 Q96RJ0 3/20 0.59
CHRNB2 P17787 1/20 0.55
CHRNA4 P43681 1/20 0.55
PTGS2 P35354 5/20 0.47
KIF11 P52732 1/20 0.46
CCR2 P41597 1/20 0.45
GRIN2B Q13224 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8604439 0.81 PTGS2 (0.52) PTGS2CCR2
SCHEMBL5811040 0.81 PTGS2 (0.50) PTGS2CA12CA1CA2CA9
SCHEMBL29113143 0.80 PTGS2 (0.53) PTGS2CCR2
Ammonia Solution, Strong SCHEMBL28859730 0.80 HTR2A (0.57) HTR2ATAAR1CHRNB2CHRNA4CA12
SCHEMBL4975056 0.79 PTGS2 (0.44) PTGS2CCR2
SCHEMBL4977528 0.79 PTGS2 (0.44) PTGS2CCR2
SCHEMBL6011425 0.79 CCR2 (0.49) PTGS2CCR2
SCHEMBL4976401 0.79 CCR2 (0.49) PTGS2CCR2
SCHEMBL17069339 0.79 PTGS2 (0.52) PTGS2
SCHEMBL30395150 0.79 PTGS2 (0.52) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5723489-A ADRENERGIC BLOCKING AGENTS OR STIMULANTS FOR GASTROINTESTINAL DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-03-03 US disclosed