SCHEMBL8606262

SCHEMBL8606262

COc1ccc2c(OC(C)=O)cn(C(=O)c3ccc(Cl)cc3)c2c1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 12/20 0.55
AKR1C2 P52895 9/20 0.55
PTGS1 P23219 2/20 0.55
AKR1C4 P17516 1/20 0.55
ABCB1 P08183 1/20 0.49
POLB P06746 2/20 0.47
AR P10275 1/20 0.47
KMT2A Q03164 2/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8606141 0.86 AKR1C3 (0.47) AKR1C3AKR1C2PTGS1AKR1C4POLB
SCHEMBL8605079 0.84 PTGS1 (0.46) AKR1C3AKR1C2PTGS1AKR1C4POLB
SCHEMBL8604032 0.81 AKR1C3 (0.47) AKR1C3AKR1C2PTGS1AKR1C4ABCB1
SCHEMBL8606260 0.78 AKR1C3 (0.83) AKR1C3AKR1C2PTGS1AKR1C4ABCB1
SCHEMBL21578435 0.76 AKR1C3 (0.70) AKR1C3AKR1C2PTGS1AKR1C4ABCB1
SCHEMBL8604631 0.76 PTGS1 (0.41) AKR1C3AKR1C2PTGS1AKR1C4ABCB1
SCHEMBL8603649 0.76 ABCB1 (0.65) AKR1C3AKR1C2PTGS1AKR1C4ABCB1
SCHEMBL3241798 0.76 ABCB11 (0.46) POLBKMT2AMAPTHPGD
SCHEMBL6271277 0.75 AKR1C3 (0.54) AKR1C3AKR1C2PTGS1AKR1C4AR
SCHEMBL8602252 0.75 KMT2A (0.48) AKR1C3AKR1C2PTGS1AKR1C4ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721347-A Esters and amides of substituted pyrrole acetic acids CELL PATHWAYS, INC. (US) 1998-02-24 US disclosed
EP-0485157-A2 Esters and amides of substituted pyrrole acetic acids FGN, INC. (US) 1992-05-13 EP disclosed