SCHEMBL8610016

SCHEMBL8610016

OP(c1cc(F)cc(F)c1)c1cc(F)cc(F)c1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA9 Q16790 1/20 0.45
CES2 O00748 2/20 0.39
CES1 P23141 2/20 0.39
IDO1 P14902 2/20 0.35
RAPGEF4 Q8WZA2 1/20 0.30
NOTUM Q6P988 1/20 0.30
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12621192 0.81 CA12 (0.45) CA12CA1CA9CES2CES1
SCHEMBL1506225 0.73 CA12 (0.42) CA12CA1CA9CES2CES1
SCHEMBL449836 0.71
SCHEMBL19968355 0.69 CA12 (0.38) CA12CA1CA9CES2CES1
SCHEMBL8059616 0.69 ORAI1 (0.39) CA1CA9CES2CES1IDO1
SCHEMBL8019916 0.69 CA12 (0.38) CA12CA1CA9CES2CES1
SCHEMBL8609628 0.69 CES2 (0.39) CA12CA1CA9CES2CES1
SCHEMBL2881917 0.69 CA12 (0.38) CA12CA1CA9CES2CES1
Methyl Alcohol SCHEMBL27837464 0.68 CA9 (0.60) CA12CA1CA9CES2CES1
SCHEMBL6250580 0.67 CA12 (0.36) CA12CA1CA9CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832087-A1 SYNTHESIS OF AND HYDROFORMYLATION WITH FLUORO-SUBSTITUTED BIDENTATE PHOSPHINE LIGANDS HOECHST CELANESE CORPORATION (US) 1998-04-01 EP claimed
US-5616785-A BIS/3,5-DIFLUOROPHENYL/PHOSPHINE OXIDE AND BIS/3,5-DIFLUOROPHENYL/-PHOSPHINOUS ACID; CHEMICAL INTERMEDIATES FOR FLUORO-SUBSTITUTED BIDENTATE PHOSPHINE LIGANDS HOECHST CELANESE CORPORATION (US) 1997-04-01 US claimed
WO-1996038456-A1 SYNTHESIS OF AND HYDROFORMYLATION WITH FLUORO-SUBSTITUTED BIDENTATE PHOSPHINE LIGANDS HOECHST CELANESE CORPORATION (US) 1996-12-05 WO claimed
EP-0739333-B1 SELECTIVE ASYMMETRIC HYDROGENATION OF DEHYDROAMINO ACID DERIVATIVES USING RHODIUM AND IRIDIUM DIPHOSPHINITE CARBOHYDRATE CATALYST COMPOSITIONS DU PONT (US) 1998-10-14 EP disclosed
US-5789624-A HYDROFORMYLATION OF ALKENES TO ALDEHYDES USING A RHODIUM COMPLEX CATALYST HOECHST CELANESE CORPORATION (US) 1998-08-04 US disclosed
US-5773661-A REACTION OF ALKALI METAL PHOSPHIDE WITH DISULFONIC ACID ESTEROF TRANS-2,3-NOBORNANEDIMETHANOL CELANESE INTERNATIONAL CORPORATION (US) 1998-06-30 US disclosed
EP-0832087-A1 SYNTHESIS OF AND HYDROFORMYLATION WITH FLUORO-SUBSTITUTED BIDENTATE PHOSPHINE LIGANDS HOECHST CELANESE CORPORATION (US) 1998-04-01 EP disclosed
US-5710338-A FLUOROPHENYLPHOSPHINE LIGANDS FOR CATALYSTS HOECHST CELANESE CORPORATION (US) 1998-01-20 US disclosed
US-5710337-A RHODIUM COMPLEX OF BIS PHOSPHINE HOECHST CELANESE CORPORATION (US) 1998-01-20 US disclosed
US-5616785-A BIS/3,5-DIFLUOROPHENYL/PHOSPHINE OXIDE AND BIS/3,5-DIFLUOROPHENYL/-PHOSPHINOUS ACID; CHEMICAL INTERMEDIATES FOR FLUORO-SUBSTITUTED BIDENTATE PHOSPHINE LIGANDS HOECHST CELANESE CORPORATION (US) 1997-04-01 US disclosed
WO-1996038456-A1 SYNTHESIS OF AND HYDROFORMYLATION WITH FLUORO-SUBSTITUTED BIDENTATE PHOSPHINE LIGANDS HOECHST CELANESE CORPORATION (US) 1996-12-05 WO disclosed
EP-0739333-A1 SELECTIVE ASYMMETRIC HYDROGENATION OF DEHYDROAMINO ACID DERIVATIVES USING RHODIUM AND IRIDIUM DIPHOSPHINITE CARBOHYDRATE CATALYST COMPOSITIONS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1996-10-30 EP disclosed
US-5567856-A USING A RHODIUM COMPLEX CATALYST HOECHST CELANESE CORPORATION (US) 1996-10-22 US disclosed
US-5510507-A COORDINATION CATALYSTS; EFFICIENT ENANTIOSELECTIVITY E. I. DU PONT DE NEMOURS AND COMPANY (US) 1996-04-23 US disclosed
US-5481006-A PREPARATION OF INTERMEDIATES FOR PHARMACEUTICALS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1996-01-02 US disclosed
WO-1995018787-A1 SELECTIVE ASYMMETRIC HYDROGENATION OF DEHYDROAMINO ACID DERIVATIVES USING RHODIUM AND IRIDIUM DIPHOSPHINITE CARBOHYDRATE CATALYST COMPOSITIONS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1995-07-13 WO disclosed