SCHEMBL8610308

SCHEMBL8610308

COc1ccccc1N1CCN(CC(O)COc2ccc(C)cc2NC(C)=O)CC1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.72
KMT2A Q03164 4/20 0.72
MAPT P10636 7/20 0.68
TP53 P04637 2/20 0.68
ABCB1 P08183 8/20 0.61
ALDH1A1 P00352 2/20 0.59
LMNA P02545 4/20 0.59
MAPK1 P28482 2/20 0.59
TDP1 Q9NUW8 2/20 0.59
KDM4E B2RXH2 2/20 0.59
HIF1A Q16665 2/20 0.59
NR1I2 O75469 1/20 0.59
NR3C1 P04150 1/20 0.59
ADRB1 P08588 1/20 0.59
HTR1A P08908 1/20 0.59
ADRA2A P08913 1/20 0.59
DRD2 P14416 1/20 0.59
ADRA2B P18089 1/20 0.59
ADRA2C P18825 1/20 0.59
DRD1 P21728 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8614094 0.93 MEN1 (0.69) MEN1KMT2AMAPTTP53ABCB1
SCHEMBL8615117 0.91 MAPT (0.66) MEN1KMT2AMAPTTP53ABCB1
SCHEMBL8609331 0.83 MAPT (0.66) MEN1KMT2AMAPTTP53ABCB1
SCHEMBL8645443 0.83 ABCB1 (0.73) ABCB1
SCHEMBL9410209 0.81 MAPT (1.00) MEN1KMT2AMAPTTP53ABCB1
SCHEMBL8615289 0.81 MAPT (0.63) MEN1KMT2AMAPTTP53ABCB1
SCHEMBL8611715 0.81 HSP90AB1 (0.58) MEN1KMT2AMAPTTP53ABCB1
Hydrochloric Acid SCHEMBL9410218 0.80 MAPT (0.98) MEN1KMT2AMAPTTP53ABCB1
SCHEMBL8609924 0.80 MAPT (0.62) MEN1KMT2AMAPTTP53ABCB1
SCHEMBL11194101 0.80 ABCB1 (0.66) MEN1KMT2AABCB1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0833639-A1 PHENOXY PIPERAZINE DERIVATIVES FOR TREATING DISORDERS OF THE DOPAMINE SYSTEM F. HOFFMANN-LA ROCHE AG (CH) 1998-04-08 EP disclosed
US-5614526-A IN TREATING DISORDERS OF THE DOPAMINE SYSTEM HOFFMANN-LA ROCHE INC. (US) 1997-03-25 US disclosed
WO-1996041630-A1 PHENOXY PIPERAZINE DERIVATIVES FOR TREATING DISORDERS OF THE DOPAMINE SYSTEM F. HOFFMANN-LA ROCHE AG (CH) 1996-12-27 WO disclosed