SCHEMBL8611715

SCHEMBL8611715

CC(=O)Nc1ccccc1OCC(O)CN1CCN(c2ccccc2O)CC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 1/20 0.58
ABCB1 P08183 13/20 0.58
CCR1 P32246 2/20 0.54
MAPT P10636 3/20 0.52
ALDH1A1 P00352 2/20 0.52
LMNA P02545 2/20 0.52
MAPK1 P28482 2/20 0.52
TDP1 Q9NUW8 2/20 0.52
NR1I2 O75469 1/20 0.52
NR3C1 P04150 1/20 0.52
ADRB1 P08588 1/20 0.52
HTR1A P08908 1/20 0.52
ADRA2A P08913 1/20 0.52
DRD2 P14416 1/20 0.52
ADRA2B P18089 1/20 0.52
ADRA2C P18825 1/20 0.52
DRD1 P21728 1/20 0.52
ACHE P22303 1/20 0.52
SLC6A2 P23975 1/20 0.52
HRH2 P25021 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8615117 0.90 MAPT (0.66) HSP90AB1ABCB1MAPTALDH1A1LMNA
SCHEMBL8645443 0.90 ABCB1 (0.73) ABCB1
SCHEMBL8613687 0.86 HSP90AB1 (0.55) HSP90AB1ABCB1CCR1KCNH2
SCHEMBL8609331 0.82 MAPT (0.66) ABCB1MAPTALDH1A1LMNAMAPK1
SCHEMBL8614094 0.81 MEN1 (0.69) ABCB1MAPTALDH1A1LMNAMAPK1
SCHEMBL8610308 0.81 MEN1 (0.72) ABCB1MAPTALDH1A1LMNAMAPK1
SCHEMBL11818605 0.80 HSP90AB1 (0.57) HSP90AB1ABCB1MAPTLMNAMAPK1
SCHEMBL8615289 0.80 MAPT (0.63) ABCB1MAPTALDH1A1LMNAMAPK1
SCHEMBL8637503 0.80 ABCB1 (0.60) ABCB1MAPTALDH1A1LMNAMAPK1
Hydrochloric Acid SCHEMBL11816206 0.80 HSP90AB1 (0.56) HSP90AB1ABCB1MAPTALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0833639-A1 PHENOXY PIPERAZINE DERIVATIVES FOR TREATING DISORDERS OF THE DOPAMINE SYSTEM F. HOFFMANN-LA ROCHE AG (CH) 1998-04-08 EP disclosed
US-5614526-A IN TREATING DISORDERS OF THE DOPAMINE SYSTEM HOFFMANN-LA ROCHE INC. (US) 1997-03-25 US disclosed
WO-1996041630-A1 PHENOXY PIPERAZINE DERIVATIVES FOR TREATING DISORDERS OF THE DOPAMINE SYSTEM F. HOFFMANN-LA ROCHE AG (CH) 1996-12-27 WO disclosed