SCHEMBL8610309

SCHEMBL8610309

CS(=O)(=O)c1ccc(-n2nc(C(F)(F)F)cc2-c2ccccc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 11/20 1.00
PTGS1 P23219 3/20 0.79
CYP2C9 P11712 1/20 0.79
PDPK1 O15530 1/20 0.73
ALOX5 P09917 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8765387 0.95 PTGS2 (0.90) PTGS2PTGS1CYP2C9PDPK1ALOX5
SCHEMBL9260744 0.90 PTGS2 (0.81) PTGS2PTGS1CYP2C9PDPK1ALOX5
SCHEMBL9257388 0.90 PTGS2 (0.81) PTGS2PTGS1CYP2C9PDPK1ALOX5
SCHEMBL6957077 0.90 PTGS2 (0.80) PTGS2PTGS1CYP2C9PDPK1ALOX5
SCHEMBL9088072 0.90 PTGS2 (0.80) PTGS2PTGS1CYP2C9PDPK1
SCHEMBL5229949 0.88 PTGS2 (1.00) PTGS2PTGS1CYP2C9PDPK1ALOX5
Sc-58125 SCHEMBL214120 0.88 PTGS2 (1.00) PTGS2PTGS1CYP2C9PDPK1ALOX5
SCHEMBL6378189 0.88 PTGS2 (1.00) PTGS2PTGS1CYP2C9PDPK1ALOX5
SCHEMBL8953888 0.88 PTGS2 (1.00) PTGS2PTGS1CYP2C9PDPK1ALOX5
SCHEMBL8954103 0.88 PTGS2 (0.81) PTGS2PTGS1CYP2C9PDPK1ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0830133-A1 THERAPEUTIC COMPOSITION FOR ARTHRITIS Takeda Chemical Industries, Ltd. (JP) 1998-03-25 EP disclosed
WO-1996033717-A1 THERAPEUTIC COMPOSITION FOR ARTHRITIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-10-31 WO disclosed
US-5475018-A Antiinflammatory agent, antiarthritic agent; analgesics and antipyretics G. D. SEARLE & CO. (US) 1995-12-12 US disclosed