SCHEMBL9260744

SCHEMBL9260744

CS(=O)(=O)c1ccc(-n2nc(C(F)(F)Cl)cc2-c2ccccc2)cc1

nearest known ligand 0.81

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.81
ALOX5 P09917 2/20 0.67
PTGS1 P23219 3/20 0.65
CYP2C9 P11712 1/20 0.65
PDPK1 O15530 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8610309 0.90 PTGS2 (1.00) PTGS2ALOX5PTGS1CYP2C9PDPK1
SCHEMBL8640401 0.89 PTGS2 (0.82) PTGS2PTGS1CYP2C9
SCHEMBL9003005 0.89 PTGS2 (0.67) PTGS2PTGS1CYP2C9PDPK1
SCHEMBL9003167 0.88 PTGS2 (0.65) PTGS2PTGS1CYP2C9
SCHEMBL9002935 0.88 PTGS2 (0.82) PTGS2ALOX5PTGS1CYP2C9PDPK1
SCHEMBL9257388 0.88 PTGS2 (0.81) PTGS2ALOX5PTGS1CYP2C9PDPK1
SCHEMBL9003059 0.85 PTGS2 (0.78) PTGS2ALOX5PTGS1CYP2C9PDPK1
SCHEMBL8765387 0.85 PTGS2 (0.90) PTGS2ALOX5PTGS1CYP2C9PDPK1
SCHEMBL17369546 0.80 ALOX5 (1.00) PTGS2ALOX5PTGS1CYP2C9
SCHEMBL6957077 0.80 PTGS2 (0.80) PTGS2ALOX5PTGS1CYP2C9PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5475018-A Antiinflammatory agent, antiarthritic agent; analgesics and antipyretics G. D. SEARLE & CO. (US) 1995-12-12 US disclosed