SCHEMBL8610558

SCHEMBL8610558

CC(=O)Nc1cc(N)c(Cl)cc1NC(C)=O

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
HDAC1 Q13547 3/20 0.45
HDAC3 O15379 2/20 0.45
HDAC2 Q92769 2/20 0.45
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 1/20 0.43
HSD17B10 Q99714 1/20 0.43
GAA P10253 2/20 0.42
NPC1 O15118 2/20 0.41
PGK1 P00558 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40
ROCK2 O75116 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11069418 0.90 CA1 (0.50) CA1CA2CA9HDAC1HDAC3
SCHEMBL9137511 0.90 CA1 (0.50) CA1CA2CA9HDAC1HDAC3
SCHEMBL8777806 0.87 CA1 (0.44) CA1CA2CA9HDAC1HDAC3
Butanedione SCHEMBL28088921 0.87 CA1 (0.47) CA1CA2CA9HDAC1HDAC3
SCHEMBL6811137 0.87 POLB (0.49) CA1CA2CA9HDAC1HDAC3
SCHEMBL6815913 0.87 CA1 (0.44) CA1CA2CA9HDAC1HDAC3
SCHEMBL6202482 0.85 CA1 (0.46) CA1CA2CA9HDAC1HDAC3
SCHEMBL11640102 0.85 CA1 (0.47) CA1CA2CA9HDAC1HDAC3
SCHEMBL29904715 0.84 HDAC1 (0.49) CA1CA2CA9HDAC1HDAC3
SCHEMBL1143315 0.84 HDAC1 (0.49) CA1CA2CA9HDAC1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852017-A 2,3(1H,4H)-quinoxalinediones BASF AKTIENGESELLSCHAFT (DE) 1998-12-22 US disclosed
EP-0572852-B1 Quinoxalin-2,3(1H,4H)-diones used as medicine BASF AG (DE) 1998-10-21 EP disclosed
US-5714489-A 2,3(1H,4H)quinoxalinedione BASF AKTIENGESELLSCHAFT (DE) 1998-02-03 US disclosed
EP-0572852-A1 Quinoxalin-2,3(1H,4H)-diones used as medicine BASF Aktiengesellschaft (DE) 1993-12-08 EP disclosed