SCHEMBL8611205

SCHEMBL8611205

O=C(c1nccn1C1CCCCC1)c1nccn1C1CCCCC1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.42
PDE4B Q07343 1/20 0.41
PDE4D Q08499 1/20 0.41
HSD17B10 Q99714 1/20 0.40
GAA P10253 1/20 0.40
ALDH1A1 P00352 2/20 0.40
NPC1 O15118 1/20 0.40
HPGD P15428 1/20 0.40
TP53 P04637 4/20 0.38
THRB P10828 2/20 0.38
CNOT7 Q9UIV1 1/20 0.36
HCAR1 Q9BXC0 3/20 0.36
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27700737 0.86 LMNA (0.40) LMNAPDE4BPDE4DHSD17B10GAA
SCHEMBL28416472 0.86 LMNA (0.45) LMNAPDE4BPDE4DHSD17B10GAA
SCHEMBL2364931 0.84 LMNA (0.41) LMNAPDE4BPDE4DHSD17B10GAA
SCHEMBL25601807 0.82 LMNA (0.42) LMNAPDE4BPDE4DHSD17B10GAA
SCHEMBL28411151 0.78 LMNA (0.38) LMNAPDE4BPDE4DHSD17B10GAA
SCHEMBL30554006 0.77 ALDH1A1 (0.43) LMNAGAAALDH1A1NPC1HPGD
SCHEMBL30554033 0.73 ALDH1A1 (0.40) LMNAHSD17B10GAAALDH1A1NPC1
SCHEMBL9442396 0.72 PI4KA (0.37) LMNAHSD17B10GAAALDH1A1NPC1
SCHEMBL3237878 0.72 PI4KA (0.37) LMNAHSD17B10GAATP53THRB
SCHEMBL4964108 0.72 KDM4E (0.40) LMNAGAATHRBHCAR1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5770701-A Process for preparing targeted forms of methyltrithio antitumor agents AMERICAN CYANAMID COMPANY (US) 1998-06-23 US disclosed
EP-0313873-B1 Targeted forms of methyltrithio antitumor agents AMERICAN CYANAMID CO (US) 1994-09-28 EP disclosed
EP-0313874-B1 Disulfur analogs of LL-E33288 antitumor agents AMERICAN CYANAMID CO (US) 1994-04-13 EP disclosed
US-5053394-A Protein-drug reaction product AMERICAN CYANAMID COMPANY (US) 1991-10-01 US disclosed
EP-0392384-A2 Targeted forms of methyltrithio antitumor agents AMERICAN CYANAMID COMPANY (US) 1990-10-17 EP disclosed
EP-0313873-A1 Targeted forms of methyltrithio antitumor agents AMERICAN CYANAMID COMPANY (US) 1989-05-03 EP disclosed
EP-0313874-A2 Disulfur analogs of LL-E33288 antitumor agents AMERICAN CYANAMID COMPANY (US) 1989-05-03 EP disclosed