SCHEMBL8611247

SCHEMBL8611247

CC=C(c1ccccc1)C(c1ccccc1)c1ccc(OCCN)cc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 13/20 0.51
ESR1 P03372 10/20 0.51
ESR2 Q92731 10/20 0.51
CYP3A4 P08684 2/20 0.51
TAAR1 Q96RJ0 1/20 0.50
LTA4H P09960 2/20 0.49
PLA2G2A P14555 1/20 0.49
CYP1A2 P05177 1/20 0.47
CYP2A6 P11509 1/20 0.47
CYP3A5 P20815 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
ALDH1A1 P00352 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7032426 1.00 CYP19A1 (0.51) CYP19A1ESR1ESR2CYP3A4TAAR1
SCHEMBL4620169 0.89 GAA (0.51) CYP19A1ESR1ESR2CYP3A4LTA4H
SCHEMBL10893461 0.87 ALDH1A1 (0.41) CYP19A1ESR1ESR2CYP3A4LTA4H
SCHEMBL11266486 0.87 ALDH1A1 (0.44) CYP19A1ESR1ESR2CYP3A4LTA4H
SCHEMBL2710225 0.85 CYP2D6 (0.55) ESR1ESR2CYP3A4LTA4HCYP1A2
SCHEMBL8732737 0.85 CYP2D6 (0.55) ESR1ESR2CYP3A4LTA4HCYP1A2
SCHEMBL7929087 0.85 CYP2D6 (0.55) ESR1ESR2CYP3A4LTA4HCYP1A2
SCHEMBL11377599 0.82 ALDH1A1 (0.46) TAAR1SMN1; SMN2ALDH1A1NPSR1
SCHEMBL9661912 0.81 ESR1 (0.47) CYP19A1ESR1ESR2CYP3A4CYP1A2
SCHEMBL11482997 0.80 KMT2A (0.44) CYP1A2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729363-A4 BORON-CONTAINING HORMONE ANALOGS AND METHODS OF THEIR USE IN IMAGING OR KILLING CELLS HAVING HORMONE RECEPTORS IONIX CORP (US) 1998-08-19 EP disclosed
EP-0729363-A1 BORON-CONTAINING HORMONE ANALOGS AND METHODS OF THEIR USE IN IMAGING OR KILLING CELLS HAVING HORMONE RECEPTORS IONIX CORPORATION (US) 1996-09-04 EP disclosed
WO-1996000090-A1 BORON-CONTAINING HORMONE ANALOGS AND METHODS OF THEIR USE IN IMAGING OR KILLING CELLS HAVING HORMONE RECEPTORS IONIX CORPORATION (US) 1996-01-04 WO disclosed