SCHEMBL8612754

SCHEMBL8612754

Nc1nc(N)c2ncn([C@@H]3O[C@H](COC(c4ccccc4)(c4ccccc4)c4ccccc4)[C@@H](O)[C@H]3O)c2n1

nearest known ligand 0.67

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TYMP P19971 10/20 0.67
ADORA1 P30542 2/20 0.67
HINT1 P49773 2/20 0.66
NT5E P21589 2/20 0.61
ADORA2A P29274 2/20 0.57
ADORA2B P29275 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8612666 0.91 TYMP (0.56) TYMPADORA1HINT1NT5EADORA2A
SCHEMBL8610421 0.91 TYMP (0.56) TYMPADORA1HINT1NT5E
SCHEMBL8610725 0.91 NT5E (0.66) TYMPADORA1HINT1NT5EADORA2A
SCHEMBL8610719 0.91 TYMP (0.75) TYMPADORA1HINT1NT5E
SCHEMBL8614413 0.88 SLC29A1 (0.63) TYMPADORA1
SCHEMBL10834193 0.88 ADORA1 (0.62) TYMPADORA1HINT1NT5EADORA2A
SCHEMBL8614976 0.88 TYMP (0.62) TYMPADORA1HINT1
SCHEMBL8610899 0.87 ADORA1 (0.82) TYMPADORA1ADORA2AADORA2B
SCHEMBL31484253 0.87 ADORA1 (0.82) TYMPADORA1ADORA2AADORA2B
SCHEMBL8610903 0.87 ADORA1 (0.82) TYMPADORA1ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992011276-A1 NOVEL SYNTHESIS OF 2'-'UP' FLUORINATED 2''-DEOXY-ARABINOFURANOSYLPURINES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-07-09 WO claimed
US-5750675-A 2'-\"up\" fluorinated 2'-deoxy-arabinofuranosylpurines SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1998-05-12 US disclosed
US-5525720-A Synthesis of 2'-\"up\" fluorinated 2'-deoxy-arabinofuranosyl purines SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1996-06-11 US disclosed
WO-1992011276-A1 NOVEL SYNTHESIS OF 2'-'UP' FLUORINATED 2''-DEOXY-ARABINOFURANOSYLPURINES SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1992-07-09 WO disclosed