SCHEMBL8613565

SCHEMBL8613565

COc1ccc(CCNCC(O)CN2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1OC

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 8/20 0.63
LMNA P02545 3/20 0.61
OXTR P30559 1/20 0.61
AVPR1A P37288 1/20 0.61
HTT P42858 1/20 0.61
ADRB1 P08588 7/20 0.56
ADRB3 P13945 5/20 0.56
ALDH1A1 P00352 2/20 0.51
SLC6A4 P31645 2/20 0.51
SLC6A3 Q01959 2/20 0.51
NPSR1 Q6W5P4 1/20 0.51
SLC22A1 O15245 1/20 0.51
CHRM2 P08172 1/20 0.51
CYP3A4 P08684 1/20 0.51
CHRM1 P11229 1/20 0.51
TSHR P16473 1/20 0.51
NFKB1 P19838 1/20 0.51
OPRM1 P35372 1/20 0.51
HIF1A Q16665 1/20 0.51
HTR1A P08908 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9416469 0.94 ADRB2 (0.57) ADRB2LMNAOXTRAVPR1AHTT
SCHEMBL8616198 0.85 CCR3 (0.53) ADRB2LMNAHTTALDH1A1NPSR1
SCHEMBL24322660 0.84 MEN1 (0.58) ALDH1A1NPSR1OPRM1KCNH2MEN1
SCHEMBL8612921 0.84 MEN1 (0.58) ALDH1A1NPSR1OPRM1KCNH2MEN1
SCHEMBL9147179 0.82 KMT2A (0.48) HTTALDH1A1OPRM1KCNH2GAA
Hydrochloric Acid SCHEMBL31650952 0.80 HTT (0.69) LMNAHTTALDH1A1TSHRGAA
SCHEMBL11257835 0.78 ADRB2 (1.00) ADRB2LMNAOXTRAVPR1AHTT
Tamolarizine SCHEMBL331314 0.77 KMT2A (0.67) ADRB2LMNAHTTADRB1ADRB3
Tamolarizine SCHEMBL29352586 0.76 MEN1 (0.65) ADRB2ADRB1ADRB3ALDH1A1OPRM1
Tamolarizine SCHEMBL2194434 0.76 MEN1 (0.65) ADRB2ADRB1ADRB3ALDH1A1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0549796-B1 DIPHENYLPIPERAZINE DERIVATIVE AND DRUG FOR CIRCULATORY ORGAN CONTAINING THE SAME POLA CHEM IND INC (JP) 1998-04-29 EP disclosed
US-5391552-A Has strong antagonism against calcium with less side effects POLA CHEMICAL INDUSTRIES, INC. (JP) 1995-02-21 US disclosed
EP-0612738-A1 Diphenylpiperazine derivative and drug for circulatory organ containing the same POLA CHEMICAL INDUSTRIES, INC. (JP) 1994-08-31 EP disclosed
EP-0549796-A1 DIPHENYLPIPERAZINE DERIVATIVE AND DRUG FOR CIRCULATORY ORGAN CONTAINING THE SAME POLA CHEMICAL INDUSTRIES INC (JP) 1993-07-07 EP disclosed