SCHEMBL8613877

SCHEMBL8613877

Fc1cc(OCc2ccccc2)ccc1-c1ccc(-c2cccc(F)c2F)c(F)c1F

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.51
TOP1 P11387 1/20 0.48
PDK2 Q15119 1/20 0.47
MAOB P27338 6/20 0.47
MAOA P21397 3/20 0.47
GRM5 P41594 1/20 0.45
FFAR1 O14842 1/20 0.44
LCK P06239 1/20 0.43
CYP3A4 P08684 1/20 0.43
GSTP1 P09211 1/20 0.43
CYP4F2 P78329 1/20 0.43
CYP4A11 Q02928 1/20 0.43
BCHE P06276 1/20 0.43
MRGPRX4 Q96LA9 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8616565 0.99 ALOX5 (0.53) ALOX5TOP1PDK2MAOBMAOA
SCHEMBL8617314 0.92 FFAR1 (0.49) ALOX5TOP1PDK2MAOBMAOA
SCHEMBL8612218 0.91 FFAR1 (0.47) ALOX5TOP1PDK2MAOBMAOA
SCHEMBL8612975 0.89 GSTP1 (0.51) ALOX5TOP1PDK2MAOBMAOA
SCHEMBL8612830 0.88 GSTP1 (0.50) ALOX5MAOBGRM5FFAR1GSTP1
SCHEMBL8611289 0.86 GSTP1 (0.54) ALOX5MAOBMAOAGRM5FFAR1
SCHEMBL8612316 0.84 ALOX5 (0.50) ALOX5TOP1PDK2MAOBMAOA
SCHEMBL8615452 0.84 MAOB (0.55) ALOX5TOP1PDK2MAOBMAOA
SCHEMBL8612910 0.84 ALOX5 (0.50) ALOX5TOP1PDK2MAOBMAOA
SCHEMBL8613886 0.84 FFAR1 (0.47) ALOX5TOP1MAOBMAOAFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0665836-B1 BIFUNCTIONAL INTERMEDIATES FOR USE IN THE MANUFACTURE OF LIQUID CRYSTALS HOECHST AG (DE) 1998-04-29 EP disclosed
WO-1994010152-A1 BIFUNCTIONAL INTERMEDIATES FOR USE IN THE MANUFACTURE OF LIQUID CRYSTALS HOECHST AKTIENGESELLSCHAFT (DE) 1994-05-11 WO disclosed