SCHEMBL8613890

SCHEMBL8613890

CC(=O)C(C)CC(C)C#N

nearest known ligand 0.38

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.36
CHRM1 P11229 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8534653 0.81 NAALAD2 (0.43) TSHR
SCHEMBL18768867 0.79 CHRM1 (0.32) CHRM1
SCHEMBL9575752 0.77 TSHR (0.33) TSHR
SCHEMBL17953984 0.76 ALDH1A1 (0.40) CHRM1
SCHEMBL12891365 0.76 ALDH1A1 (0.40) CHRM1
SCHEMBL19233793 0.76 SMN1; SMN2 (0.35) TSHR
SCHEMBL15092131 0.73 TSHR (0.37) TSHR
SCHEMBL9753145 0.73 TSHR (0.33) TSHR
SCHEMBL24486625 0.73 HDAC7 (0.41) TSHRCHRM1
SCHEMBL12050688 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0437290-B1 Process for the preparation of 5-oxohexane nitriles and the compound 2,4-dimethyl-5-oxohexane nitrile DSM NV (NL) 1998-05-06 EP claimed
US-5334721-A Reacting a methyl ketone and an alpha,beta-unsaturated nitrile in the presence of a basic catalyst; preparation of a 2-methyl-3,5-dialkylpyridine; cyclization; dehydrogenation STAMICARBON B.V. (NL) 1994-08-02 US claimed
US-5254712-A Using basic catalyst STAMICARBON B.V. (NL) 1993-10-19 US claimed
EP-0437290-A1 Process for the preparation of 5-oxohexane nitriles and the compound 2,4-dimethyl-5-oxohexane nitrile DSM N.V. (NL) 1991-07-17 EP claimed
JP-4253946-A None JP disclosed
EP-2032989-B2 IGFBP2 BIOMARKER MERCK SHARP & DOHME (US) 2015-10-28 EP disclosed
EP-0437290-B1 Process for the preparation of 5-oxohexane nitriles and the compound 2,4-dimethyl-5-oxohexane nitrile DSM NV (NL) 1998-05-06 EP disclosed
EP-0437290-B1 Process for the preparation of 5-oxohexane nitriles and the compound 2,4-dimethyl-5-oxohexane nitrile DSM NV (NL) 1998-05-06 EP disclosed
US-5334721-A Reacting a methyl ketone and an alpha,beta-unsaturated nitrile in the presence of a basic catalyst; preparation of a 2-methyl-3,5-dialkylpyridine; cyclization; dehydrogenation STAMICARBON B.V. (NL) 1994-08-02 US disclosed
US-5334721-A Reacting a methyl ketone and an alpha,beta-unsaturated nitrile in the presence of a basic catalyst; preparation of a 2-methyl-3,5-dialkylpyridine; cyclization; dehydrogenation STAMICARBON B.V. (NL) 1994-08-02 US disclosed
US-5254712-A Using basic catalyst STAMICARBON B.V. (NL) 1993-10-19 US disclosed
US-5254712-A Using basic catalyst STAMICARBON B.V. (NL) 1993-10-19 US disclosed
US-5254712-A Using basic catalyst STAMICARBON B.V. (NL) 1993-10-19 US disclosed
JP-H04253946-A PRODUCTION OF 5-OXOHEXANENITRILE,2,4-DIMETHYL-5-OXOHEXANENITRILE AND 2,3,5-TRIMETHYLPYRIDINE AND 2-METHYL-3,5-DIALKYLPYRIDINE STAMICARBON BV 1992-09-09 JP disclosed
WO-1991017979-A1 PROCESS FOR THE PREPARATION OF 2-N-ACYLAMINOPYRIDINES AND 2-AMINOPYRIDINES FROM 5-OXOALKANENITRILE OXIMES DSM N.V. (NL) 1991-11-28 WO disclosed
EP-0437290-A1 Process for the preparation of 5-oxohexane nitriles and the compound 2,4-dimethyl-5-oxohexane nitrile DSM N.V. (NL) 1991-07-17 EP disclosed
EP-0437290-A1 Process for the preparation of 5-oxohexane nitriles and the compound 2,4-dimethyl-5-oxohexane nitrile DSM N.V. (NL) 1991-07-17 EP disclosed
EP-0437290-A1 Process for the preparation of 5-oxohexane nitriles and the compound 2,4-dimethyl-5-oxohexane nitrile DSM N.V. (NL) 1991-07-17 EP disclosed