SCHEMBL8614044

SCHEMBL8614044

CCC(C)CCc1ccc2nc(-c3ccccc3)cc(C(=O)NC(=N)N)c2c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 12/20 0.46
TACR2 P21452 2/20 0.46
CA12 O43570 3/20 0.43
CA1 P00915 3/20 0.43
CA2 P00918 3/20 0.43
CA9 Q16790 3/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
RECQL P46063 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8616636 0.86 KDM4E (0.52) TACR3TACR2CA12CA1CA2
SCHEMBL8619212 0.85 DHODH (0.53) TACR3CA12CA1CA2CA9
SCHEMBL8615299 0.84 TACR3 (0.49) TACR3TACR2KDM4EALDH1A1LMNA
SCHEMBL8616486 0.83 TACR3 (0.47) TACR3TACR2CA12CA1CA2
SCHEMBL8619733 0.83 DHODH (0.58) TACR3TACR2TP53KDM4EALDH1A1
SCHEMBL8619650 0.81 TSHR (0.55) TACR3TACR2MAPTKDM4EALDH1A1
SCHEMBL8617740 0.80 TACR3 (0.51) TACR3TACR2KDM4ETSHR
SCHEMBL8616548 0.80 TACR3 (0.52) TACR3TACR2TP53KDM4EALDH1A1
SCHEMBL8614053 0.80 TP53 (0.55) TACR3TACR2TP53MAPTKDM4E
SCHEMBL8619034 0.79 DHODH (0.57) TACR3TACR2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed