SCHEMBL8615299

SCHEMBL8615299

CCC(C)Cc1ccc2c(C(=O)NC(=N)N)cc(-c3ccccc3)nc2c1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 14/20 0.49
TACR2 P21452 2/20 0.49
DHODH Q02127 1/20 0.47
KDM4E B2RXH2 2/20 0.45
MEN1 O00255 1/20 0.45
POLB P06746 1/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 2/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617740 0.93 TACR3 (0.51) TACR3TACR2DHODHKDM4EMEN1
SCHEMBL8619733 0.91 DHODH (0.58) TACR3TACR2DHODHKDM4EMEN1
SCHEMBL8619034 0.91 DHODH (0.57) TACR3TACR2DHODHKDM4EMEN1
SCHEMBL8619650 0.86 TSHR (0.55) TACR3TACR2DHODHKDM4EMEN1
SCHEMBL8614044 0.84 TACR3 (0.46) TACR3TACR2KDM4EALDH1A1LMNA
SCHEMBL8614305 0.83 GAA (0.51) TACR3TACR2KDM4EMEN1POLB
SCHEMBL8616486 0.82 TACR3 (0.47) TACR3TACR2DHODHKDM4EMEN1
SCHEMBL8619720 0.82 TACR3 (0.52) TACR3TACR2DHODHKDM4EALDH1A1
SCHEMBL8616636 0.81 KDM4E (0.52) TACR3TACR2KDM4EMEN1POLB
SCHEMBL8615123 0.80 DHODH (0.59) TACR3TACR2DHODHKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed