Biguanide

Biguanide

SCHEMBL8614065

N=C(N)NC(=N)N.O=C(O)c1cc(C(=O)O)cc(C2CCCCC2)c1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.53
ACMSD Q8TDX5 2/20 0.41
KMT2A Q03164 3/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
CREBBP Q92793 2/20 0.39
HAO1 Q9UJM8 1/20 0.39
KDM4E B2RXH2 1/20 0.38
GLA P06280 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HIF1A Q16665 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
SERPINE1 P05121 2/20 0.38
HDAC8 Q9BY41 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
HDAC1 Q13547 1/20 0.37
EGLN1 Q9GZT9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8613401 0.85 KMO (0.68) KMOACMSDKMT2AMEN1ALDH1A1
SCHEMBL27893460 0.83 KMO (0.65) KMOACMSDKMT2AMEN1ALDH1A1
SCHEMBL30912307 0.83 KMO (0.70) KMOACMSDKMT2AMEN1ALDH1A1
SCHEMBL2727410 0.78 KMO (0.58) KMOACMSDKMT2AMEN1ALDH1A1
SCHEMBL10068703 0.77 KMO (0.54) KMOACMSDKMT2AMEN1ALDH1A1
SCHEMBL184302 0.76 KMO (0.53) KMOACMSDALDH1A1CREBBPKDM4E
SCHEMBL2723391 0.76 KMO (0.56) KMOACMSDKMT2AMEN1ALDH1A1
SCHEMBL27629794 0.75 KMO (0.49) KMOACMSDKMT2AMEN1ALDH1A1
SCHEMBL10068933 0.75 KMO (0.51) KMOACMSDKMT2AALDH1A1POLB
SCHEMBL4392929 0.74 KMO (0.55) KMOACMSDALDH1A1CREBBPKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731350-A Substituted benzenedicarboxylic acid diguanides, process for their preparation, their use as a medicament or diagnostic, and medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-24 US claimed
US-5731350-A Substituted benzenedicarboxylic acid diguanides, process for their preparation, their use as a medicament or diagnostic, and medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-24 US disclosed