SCHEMBL8620892

SCHEMBL8620892

Cc1ccccc1-c1cc(NC(=N)NC=O)c2ccccc2n1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.47
MEN1 O00255 5/20 0.45
KMT2A Q03164 5/20 0.45
POLB P06746 1/20 0.45
ALDH1A1 P00352 4/20 0.43
HPGD P15428 4/20 0.43
KDM4E B2RXH2 3/20 0.43
TACR3 P29371 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
MAPT P10636 1/20 0.42
GPR55 Q9Y2T6 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
ACP1 P24666 3/20 0.41
PTGER4 P35408 1/20 0.39
GALR3 O60755 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619298 0.92 ACP1 (0.44) HTTMEN1KMT2APOLBALDH1A1
SCHEMBL8613694 0.90 ALDH1A1 (0.50) HTTMEN1KMT2APOLBALDH1A1
SCHEMBL8616273 0.90 KMT2A (0.48) HTTMEN1KMT2AALDH1A1HPGD
SCHEMBL8620107 0.89 HTT (0.37) HTTMEN1KMT2APOLBALDH1A1
SCHEMBL8614948 0.89 HTT (0.39) HTTMEN1KMT2APOLBALDH1A1
SCHEMBL8615877 0.88 PTGER4 (0.41) HTTMEN1KMT2APOLBALDH1A1
SCHEMBL8615234 0.88 HTT (0.38) HTTMEN1KMT2APOLBALDH1A1
SCHEMBL8620877 0.87 HTT (0.39) HTTMEN1KMT2APOLBALDH1A1
SCHEMBL8613901 0.87 ACP1 (0.51) HTTMEN1KMT2APOLBALDH1A1
SCHEMBL8616415 0.87 ACP1 (0.42) HTTMEN1KMT2AHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed