SCHEMBL8615048

SCHEMBL8615048

Cn1ccnc1Sc1ccc(Nc2ncc3cc(O)ccc3n2)cc1Cl

nearest known ligand 0.50

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 6/20 0.50
MAP2K1 Q02750 15/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8615598 0.89 GCK (0.40) IGF1RMAP2K1
SCHEMBL8618439 0.84 IGF1R (0.62) IGF1RMAP2K1
Hydrochloric Acid SCHEMBL8620309 0.83 IGF1R (0.61) IGF1RMAP2K1
SCHEMBL8308341 0.79 IGF1R (0.50) IGF1RMAP2K1
SCHEMBL10395308 0.74 IGF1R (0.53) IGF1RMAP2K1
SCHEMBL23434 0.73 IGF1R (0.46) IGF1RMAP2K1
SCHEMBL8615673 0.72 BRAF (0.41) IGF1RMAP2K1
SCHEMBL5254528 0.69 IGF1R (0.75) IGF1RMAP2K1
SCHEMBL4453743 0.69 IGF1R (0.75) IGF1RMAP2K1
SCHEMBL23678 0.69 IGF1R (0.44) IGF1RMAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5821246-A USEFUL AS TYROSINE KINASE INHIBITORS AND FOR THE TREATMENT OF PROLIFERATIVE DISEASES SUCH AS CANCER ZENECA LIMITED (GB) 1998-10-13 US disclosed