SCHEMBL8619720

SCHEMBL8619720

CCCC(C)Cc1cccc(-c2cc(C(=O)NC(=N)N)c3ccccc3n2)c1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 13/20 0.52
KDM4E B2RXH2 2/20 0.50
ALDH1A1 P00352 1/20 0.50
LMNA P02545 1/20 0.50
GAA P10253 1/20 0.50
HTT P42858 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
PTGER4 P35408 2/20 0.47
TACR2 P21452 2/20 0.47
TP53 P04637 1/20 0.45
DHODH Q02127 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617740 0.90 TACR3 (0.51) TACR3KDM4ETACR2DHODH
SCHEMBL8616548 0.86 TACR3 (0.52) TACR3KDM4EALDH1A1LMNAGAA
SCHEMBL8614161 0.85 LMNA (0.61) TACR3KDM4EALDH1A1LMNAGAA
SCHEMBL8619733 0.83 DHODH (0.58) TACR3KDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL8615299 0.82 TACR3 (0.49) TACR3KDM4EALDH1A1LMNATACR2
SCHEMBL8619398 0.81 TACR3 (0.59) TACR3KDM4EALDH1A1PTGER4TACR2
SCHEMBL8617743 0.80 CYP3A4 (0.65) TACR3KDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL8618943 0.79 MEN1 (0.65) TACR3KDM4EALDH1A1LMNAGAA
SCHEMBL8619034 0.79 DHODH (0.57) TACR3KDM4EALDH1A1TACR2DHODH
SCHEMBL8614314 0.79 KMT2A (0.65) TACR3KDM4EALDH1A1LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed