SCHEMBL8615748

SCHEMBL8615748

O=C(N(CCCSc1ccccn1)Cc1ccccc1)C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
MAPT P10636 3/20 0.45
KMT2A Q03164 1/20 0.45
POLB P06746 2/20 0.41
LMNA P02545 2/20 0.40
HPGD P15428 3/20 0.40
TSHR P16473 1/20 0.39
SMN1; SMN2 Q16637 6/20 0.38
NPC1 O15118 6/20 0.38
RAB9A P51151 6/20 0.38
HSD17B10 Q99714 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8614253 0.99 ALDH1A1 (0.47) ALDH1A1MAPTKMT2APOLBLMNA
SCHEMBL8621464 0.93 ALDH1A1 (0.50) ALDH1A1MAPTKMT2APOLBLMNA
SCHEMBL8619159 0.88 ALDH1A1 (0.45) ALDH1A1MAPTKMT2AHPGDSMN1; SMN2
Hydrochloric Acid SCHEMBL8620197 0.87 ALDH1A1 (0.44) ALDH1A1MAPTKMT2AHPGDSMN1; SMN2
SCHEMBL8619303 0.84 ALDH1A1 (0.51) ALDH1A1MAPTKMT2APOLBLMNA
SCHEMBL8618984 0.84 ALDH1A1 (0.54) ALDH1A1MAPTKMT2APOLBLMNA
Hydrochloric Acid SCHEMBL8620325 0.83 ALDH1A1 (0.53) ALDH1A1MAPTKMT2APOLBLMNA
SCHEMBL8614877 0.83 ALDH1A1 (0.44) ALDH1A1MAPTKMT2ALMNAHPGD
SCHEMBL8966758 0.82 CYP2C19 (0.43) ALDH1A1MAPTKMT2ALMNATSHR
Hydrochloric Acid SCHEMBL8966480 0.81 CYP2C19 (0.42) ALDH1A1MAPTKMT2ALMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5767121-A ANTIINFLAMMATORY AND -ARTHRITIC AGENTS; ANTIPYRETICS; ANALGESICS; ADHESION PROTEIN EXPRESSION AND CYCLOXYGENASE AND 5-LIPOXYGENASE INHIBITORS; IMMUNOSUPPRESSANTS AND -MODULATORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-06-16 US disclosed