Nortopsentin C

Nortopsentin C

SCHEMBL8615865

Brc1ccc2c(-c3c[nH]c(-c4c[nH]c5ccccc45)n3)c[nH]c2c1

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 3/20 0.62
ADRA1B P35368 3/20 0.62
CLK1 P49759 4/20 0.52
CDK5 Q00535 4/20 0.52
CDK5R1 Q15078 4/20 0.52
GSK3B P49841 3/20 0.52
CCNB2 O95067 2/20 0.52
CDK1 P06493 2/20 0.52
CCNB1 P14635 2/20 0.52
PRKACA P17612 2/20 0.52
PRKACG P22612 2/20 0.52
PRKACB P22694 2/20 0.52
CSNK1A1 P48729 2/20 0.52
CSNK1D P48730 2/20 0.52
CSNK1E P49674 2/20 0.52
CSNK1G2 P78368 2/20 0.52
CCNB3 Q8WWL7 2/20 0.52
CSNK1G1 Q9HCP0 2/20 0.52
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nortopsentin B SCHEMBL8615899 1.00 ADRA1A (0.62) ADRA1AADRA1BCLK1CDK5CDK5R1
Nortopsentin C SCHEMBL29489919 1.00 ADRA1A (0.62) ADRA1AADRA1BCLK1CDK5CDK5R1
Nortopsentin B SCHEMBL29489896 1.00 ADRA1A (0.62) ADRA1AADRA1BCLK1CDK5CDK5R1
Nortopsentin A SCHEMBL29489899 0.93 CLK1 (0.58) ADRA1AADRA1BCLK1CDK5CDK5R1
Nortopsentin A SCHEMBL8616377 0.93 CLK1 (0.58) ADRA1AADRA1BCLK1CDK5CDK5R1
Nortopsentin D SCHEMBL29489921 0.87 PDGFRB (0.62) CLK1CDK5CDK5R1GSK3BMEN1
SCHEMBL5443201 0.82 ADRA1A (0.65) ADRA1AADRA1BCLK1CDK5CDK5R1
SCHEMBL25034159 0.79 MEN1 (0.73) ADRA1AADRA1BCLK1CDK5CDK5R1
Bromodeoxytopsentin SCHEMBL17537615 0.78 ADRA1A (0.53) ADRA1AADRA1BCLK1CDK5CDK5R1
SCHEMBL14023555 0.75 ADRA1A (0.55) ADRA1AADRA1BMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686154-B1 NOVEL USE AS ANTI-INFLAMMATORY AGENTS FOR BIS-HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF HARBOR BRANCH OCEANOGRAPHIC (US) 1998-04-22 EP claimed