SCHEMBL8616306

SCHEMBL8616306

CC(C)C(C)(C)c1ccc2c(NC(=N)NC=O)cc(-c3ccccc3)nc2c1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.40
ABCG2 Q9UNQ0 2/20 0.40
ABCC1 P33527 1/20 0.40
TACR3 P29371 3/20 0.39
ACP1 P24666 2/20 0.39
CACNA2D1 P54289 1/20 0.36
NQO2 P16083 1/20 0.35
GSK3A P49840 1/20 0.35
GSK3B P49841 1/20 0.35
ADORA1 P30542 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619429 0.89 ABCG2 (0.44) ABCB1ABCG2ABCC1TACR3ACP1
SCHEMBL8613674 0.83 TRPV1 (0.43) ABCB1ABCG2ABCC1TACR3ACP1
SCHEMBL8615808 0.83 KDM4E (0.50) ABCB1ABCG2ABCC1TACR3ACP1
SCHEMBL8617739 0.82 ALDH1A1 (0.47) ABCB1ABCG2ABCC1TACR3ACP1
SCHEMBL8617753 0.82 ACP1 (0.51) ABCB1ABCG2ABCC1ACP1
SCHEMBL8619039 0.81 DHODH (0.46) ABCB1ABCG2ABCC1TACR3ACP1
SCHEMBL8614310 0.81 TACR3 (0.44) ABCB1ABCG2ABCC1TACR3ACP1
SCHEMBL8615210 0.81 TACR3 (0.44) ABCB1ABCG2ABCC1TACR3ACP1
SCHEMBL8619415 0.80 ABCB1 (0.47) ABCB1ABCG2ABCC1TACR3ACP1
SCHEMBL8615938 0.80 TACR3 (0.41) ABCB1ABCG2ABCC1TACR3ACP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed