SCHEMBL8616308

SCHEMBL8616308

CC(C)C(C)(C)c1ccc2c(C(=O)NC(N)=Nc3ccccc3)ccnc2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.37
SMN1; SMN2 Q16637 4/20 0.37
RAB9A P51151 4/20 0.37
ALDH1A1 P00352 2/20 0.37
NPC1 O15118 2/20 0.37
SCNN1A P37088 1/20 0.37
HPGD P15428 3/20 0.36
KDM4E B2RXH2 3/20 0.36
RECQL P46063 2/20 0.36
GMNN O75496 1/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
NFKB1 P19838 1/20 0.36
THPO P40225 1/20 0.36
STAT6 P42226 1/20 0.36
PMP22 Q01453 1/20 0.36
HIF1A Q16665 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617741 0.82 SCN2A (0.44) ADORA2ASMN1; SMN2RAB9AALDH1A1NPC1
SCHEMBL8613677 0.82 SMN1; SMN2 (0.42) ADORA2ASMN1; SMN2RAB9AALDH1A1NPC1
SCHEMBL8619044 0.81 CTSV (0.40) ADORA2ASMN1; SMN2RAB9AALDH1A1NPC1
SCHEMBL8614313 0.81 RAB9A (0.39) ADORA2ASMN1; SMN2RAB9AALDH1A1NPC1
SCHEMBL8615943 0.81 RAB9A (0.45) ADORA2ASMN1; SMN2RAB9AALDH1A1NPC1
SCHEMBL8615213 0.81 RAB9A (0.42) ADORA2ASMN1; SMN2RAB9AALDH1A1NPC1
SCHEMBL8619419 0.80 SMO (0.38) ADORA2ASMN1; SMN2RAB9AALDH1A1NPC1
SCHEMBL8619393 0.80 SMN1; SMN2 (0.46) ADORA2ASMN1; SMN2RAB9AALDH1A1NPC1
SCHEMBL8618237 0.80 ALK (0.43) ADORA2ASMN1; SMN2RAB9AALDH1A1NPC1
SCHEMBL8616502 0.80 KDM4E (0.48) SMN1; SMN2RAB9AALDH1A1NPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed