SCHEMBL8616484

SCHEMBL8616484

COc1cc(OC)c2nccc(C(=O)NC(N)=Nc3ccccc3)c2c1OC

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMO Q99835 14/20 0.49
SCN5A Q14524 2/20 0.47
SCN2A Q99250 2/20 0.47
IMPDH2 P12268 1/20 0.41
RAB9A P51151 3/20 0.40
LMNA P02545 2/20 0.40
NPC1 O15118 2/20 0.40
PSMD14 O00487 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
MITF O75030 1/20 0.39
TP53 P04637 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.39
ALDH1A1 P00352 1/20 0.38
SCNN1A P37088 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8614046 0.92 SMO (0.49) SMOSCN5ASCN2AIMPDH2RAB9A
SCHEMBL8614354 0.87 SMO (0.43) SMOSCN5ASCN2AIMPDH2RAB9A
SCHEMBL8614772 0.87 SMO (0.43) SMOSCN5ASCN2AIMPDH2RAB9A
SCHEMBL8613207 0.86 SMO (0.49) SMOSCN5ASCN2AIMPDH2RAB9A
SCHEMBL8619835 0.86 SMO (0.49) SMOSCN5ASCN2AIMPDH2RAB9A
SCHEMBL8617949 0.84 SMO (0.46) SMOSCN5ASCN2AIMPDH2RAB9A
SCHEMBL8614883 0.82 SMO (0.46) SMOSCN5ASCN2AIMPDH2RAB9A
SCHEMBL8616307 0.82 SMO (0.43) SMOSCN5ASCN2AIMPDH2RAB9A
SCHEMBL8620636 0.80 NPC1 (0.49) SMOSCN5ASCN2AIMPDH2RAB9A
SCHEMBL8617725 0.80 PDE4A (0.46) SMOIMPDH2RAB9ALMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed