SCHEMBL8616307

SCHEMBL8616307

COc1cc(OC)c2nccc(C(=O)NC(N)=Nc3ccccc3)c2c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMO Q99835 9/20 0.43
IMPDH2 P12268 1/20 0.41
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
LMNA P02545 3/20 0.40
PSMD14 O00487 1/20 0.40
SCN2A Q99250 2/20 0.40
SCN5A Q14524 1/20 0.40
AURKA O14965 2/20 0.39
RPS6KB1 P23443 2/20 0.39
PKM P14618 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 3/20 0.39
MAPT P10636 2/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
SCNN1A P37088 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617785 0.96 LMNA (0.43) SMOIMPDH2NPC1RAB9ALMNA
SCHEMBL8617725 0.86 PDE4A (0.46) SMOIMPDH2NPC1RAB9ALMNA
SCHEMBL8613207 0.86 SMO (0.49) SMOIMPDH2NPC1RAB9ALMNA
SCHEMBL8618668 0.84 SMO (0.43) SMOIMPDH2NPC1RAB9ALMNA
SCHEMBL8620947 0.83 KDM4E (0.60) NPC1RAB9ALMNASCN2AKDM4E
SCHEMBL8617943 0.83 LMNA (0.45) SMOIMPDH2NPC1RAB9ALMNA
Hydrochloric Acid SCHEMBL8615174 0.83 SMO (0.42) SMOIMPDH2NPC1RAB9ALMNA
SCHEMBL8614883 0.82 SMO (0.46) SMOIMPDH2NPC1RAB9ALMNA
SCHEMBL8620870 0.82 SRC (0.47) SMONPC1RAB9ALMNAPSMD14
SCHEMBL8616484 0.82 SMO (0.49) SMOIMPDH2NPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed