SCHEMBL8616587

SCHEMBL8616587

CC(=O)Nc1ccc(Br)c(Cl)c1Cl.Nc1ccc(-c2ccncc2)c(Cl)c1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 4/20 0.39
HDAC3 O15379 3/20 0.39
HDAC1 Q13547 3/20 0.39
RXFP1 Q9HBX9 1/20 0.36
AAK1 Q2M2I8 2/20 0.35
ADORA2B P29275 3/20 0.35
ADORA3 P0DMS8 2/20 0.35
ADORA2A P29274 2/20 0.35
ADORA1 P30542 2/20 0.35
CKS1B P61024 1/20 0.35
SKP2 Q13309 1/20 0.35
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA9 Q16790 2/20 0.34
CCNC P24863 1/20 0.34
CDK8 P49336 1/20 0.34
CCNE2 O96020 1/20 0.33
CDK4 P11802 1/20 0.33
CCND1 P24385 1/20 0.33
CCNE1 P24864 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6998722 0.85 ADORA2B (0.43) HDAC2HDAC3HDAC1ADORA2BADORA3
SCHEMBL7001806 0.77 RXFP1 (0.56) HDAC1RXFP1CA1CA2CA9
SCHEMBL6990668 0.74 MAPT (0.52) AAK1ADORA2AADORA1CCNCCDK8
SCHEMBL8616595 0.72 LMNA (0.46)
SCHEMBL26921845 0.69 RXFP1 (0.48) HDAC2HDAC3HDAC1RXFP1CA1
SCHEMBL2429572 0.68 RXFP1 (0.53) HDAC1RXFP1CA1CA2CA9
SCHEMBL8118565 0.67 JAK2 (0.44) HDAC2HDAC3HDAC1KDM4ENTRK1
SCHEMBL11279567 0.67 HDAC2 (0.74) HDAC2HDAC3HDAC1AAK1
SCHEMBL8118373 0.67 RXFP1 (0.55) RXFP1ADORA2BADORA3ADORA2AADORA1
SCHEMBL16371520 0.67 NPC1 (0.51) HDAC2HDAC3HDAC1RXFP1AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998050346-A2 ACETAMIDE AND UREA DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF CNS DISORDERS SMITHKLINE BEECHAM PLC (GB) 1998-11-12 WO disclosed