SCHEMBL8616835

SCHEMBL8616835

COCc1sc(C(C)(O)c2ccsc2)nc1C

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.34
FFAR1 O14842 1/20 0.31
CASR P41180 2/20 0.30
CDC7 O00311 1/20 0.30
DBF4 Q9UBU7 1/20 0.30
PPARD Q03181 1/20 0.30
PPARA Q07869 1/20 0.30
MEN1 O00255 1/20 0.30
GFER P55789 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8613461 0.83 SRC (0.33) CASR
SCHEMBL8616495 0.79 ALDH1A1 (0.37) KDM4ECDC7DBF4PPARDPPARA
SCHEMBL8751841 0.67 CYP1A2 (0.33)
SCHEMBL8611734 0.67 CHRM3 (0.32) KDM4E
SCHEMBL8612881 0.64 AR (0.36)
SCHEMBL8614196 0.64 ALDH1A1 (0.32) KDM4E
SCHEMBL8615946 0.64 RORC (0.36) KDM4E
SCHEMBL8613471 0.63 KDM4E (0.30) KDM4E
SCHEMBL8614886 0.62 KDM4E (0.32) KDM4E
SCHEMBL11715059 0.62 HRH2 (0.57)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731335-A NERVOUS SYSTEM DISORDERS; STROKE; ANTIISCHEMIC AGENTS; COGNITION ACTIVATORS ASTRA AKTIEBOLAG (SE) 1998-03-24 US disclosed
US-5607956-A TREATMENT OF NEURODEGENERATIVE DISORDERS SUCH AS CEREBRAL ISCHEMIA, ALZHEIMER'S DISEASE ASTRA AKTIEBOLAG (SE) 1997-03-04 US disclosed
EP-0707584-A1 NOVEL (1-HETEROAZOLYL-1-HETEROCYCLYL)ALKANE DERIVATIVES AND THEIR USE AS NEUROPROTECTIVE AGENTS Astra Aktiebolag (SE) 1996-04-24 EP disclosed
WO-1995001979-A1 NOVEL (1-HETEROAZOLYL-1-HETEROCYCLYL)ALKANE DERIVATIVES AND THEIR USE AS NEUROPROTECTIVE AGENTS ASTRA AKTIEBOLAG (SE) 1995-01-19 WO disclosed